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N-ethyl-5-methyl-N-(2-methylprop-2-en-1-yl)-4-[(prop-2-en-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
(2E)-1-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(pyridin-4-yl)prop-2-en-1-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-(hydroxymethyl)benzamide
N-[2-(dimethylamino)ethyl]-5-(quinolin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-(3-fluorophenyl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-1H-pyrazole-4-carboxamide
2-(benzyloxy)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(2-methoxyethyl)methylamine
2-methyl-4-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-imidazol-2-yl)-1,3-oxazole
3-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-3-methyl-1-[2-methyl-3-(1H-pyrrol-1-yl)phenyl]urea
N-[5-(morpholin-4-yl)pentyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
methyl 4-{[(4aR,8aS)-1-[2-(5-phenyl-4H-1,2,4-triazol-3-yl)acetyl]-decahydro-1,6-naphthyridin-6-yl]methyl}benzoate
N-(2-{7-[(2,3-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxolane-2-carboxamide
methyl 3-(6-methyl-5-{[(2E)-3-(thiophen-2-yl)prop-2-enamido]methyl}-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carbonyl)benzoate
2-({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-3-methylbutan-1-ol
2-(4-acetylphenoxy)-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]acetamide
2-[(3,5-difluorophenyl)methyl]-8-(2-hydroxypropanoyl)-2,8-diazaspiro[4.5]decan-3-one
7-(2-methoxyphenyl)-2-(phenoxymethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]-5-methyl-1,2-oxazole-3-carboxamide
methyl 1-[(3R,5S)-5-[4-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-{[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}piperidin-2-one
N-benzyl-2-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
3-{1-[2-(2H-indazol-2-yl)acetyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
2-benzyl-8-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecane
N-[(4-cyanophenyl)methyl]-2-(1-methylpiperidin-2-yl)acetamide
2-(methylsulfanyl)-7-({3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}methyl)-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
1-[(4-chlorophenyl)methyl]-4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
5-ethyl-5-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
N-methyl-2-(1-methyl-1H-pyrrol-2-yl)-2-oxo-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]acetamide
3-[4-(2-methoxyacetamido)-1H-pyrazol-1-yl]-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]benzamide
4-(2-amino-6-methylpyrimidin-4-yl)-1-[(2-fluorophenyl)methyl]piperazin-2-one
1-{4-[4-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-1-yl]phenyl}ethan-1-one
2-amino-8-[5-(1H-pyrazol-3-yl)furan-2-yl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
3-chloro-2-fluoro-N-[(1R,3S)-3-{[2-(pyridin-3-yl)ethyl]carbamoyl}cyclopentyl]benzamide
1-(1-{[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-1,4-diazepan-5-one
N-[1-(6-methylpyridin-3-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
3-chloro-N-cyclopentyl-4-({1-[(2E)-4-methylpent-2-enoyl]piperidin-4-yl}oxy)benzamide
N-(2-methoxyethyl)-5-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyridine-3-carboxamide
8-[(5-butylthiophen-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-butyl-3-(3,4-dimethyl-1H-pyrazol-5-yl)-N-(thiophen-3-ylmethyl)propanamide
4-hydroxy-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2-(thiophen-2-yl)pyrimidine-5-carboxamide
N-[2-(2-chlorophenoxy)ethyl]-4-hydroxy-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
1-{2-methoxy-5-[(4-propylpiperazin-1-yl)methyl]phenoxy}-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
2-(2-fluorophenoxymethyl)-N-methyl-N-(propan-2-yl)-1,3-oxazole-4-carboxamide
1-methyl-N-[3-(propan-2-yloxy)propyl]-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
{2-[2-(2,1,3-benzoxadiazol-5-yl)-1H-imidazol-1-yl]ethyl}diethylamine
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-propylpyrimidine-5-carboxamide
[(3S,5R)-5-[(dimethylamino)methyl]-1-{[2-(5-methylfuran-2-yl)phenyl]methyl}piperidin-3-yl]methanol
2-(dimethylamino)-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-2-(4-methylphenyl)acetamide
(2S)-1-{2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetyl}pyrrolidine-2-carboxamide