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6-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-N,N-dimethylpyrazin-2-amine
4-[2-(4-fluorophenoxy)ethyl]-1,4-oxazepan-6-ol
1-(5-methyl-1,2-oxazole-3-carbonyl)-3-(naphthalene-2-carbonyl)piperidine
5-[1-(2-methoxybenzoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
1-{1-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]piperidin-3-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
1-[3-(2-methylphenoxy)azetidin-1-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
N-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-{2-[4-(hydroxymethyl)piperidin-1-yl]ethyl}propanamide
methyl N-{2-[3-(2-chlorophenoxy)azetidin-1-yl]-2-oxoethyl}carbamate
1-[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]-2-(2-hydroxyphenyl)ethan-1-one
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
3-{1-[(2R)-2-aminopropanoyl]piperidin-4-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
2-(2,3-dihydro-1H-inden-1-yl)-1-[4-(pyrazin-2-yl)piperazin-1-yl]ethan-1-one
4-(2-methoxybenzoyl)-N-[2-(methylsulfanyl)phenyl]piperazine-1-carboxamide
9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-4-(propan-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-N'-(2-methylphenyl)-N-(1-methylpyrrolidin-3-yl)propanediamide
{2-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}urea
7-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-2-oxa-7-azaspiro[4.5]decan-8-one
3-({1-[2-methyl-3-(1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}methyl)benzoic acid
1-(4-fluorophenyl)-4-[4-(4-methyl-1H-pyrazol-3-yl)piperidin-1-yl]butane-1,4-dione
3-{4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}pyridine
1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide
4-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-carboxylic acid
1-phenyl-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperazin-2-one
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-methylpropan-1-one
2-methyl-5-({spiro[azepane-4,2'-chromene]-1-yl}carbonyl)benzene-1,3-diol
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-{[1-(morpholin-4-yl)cycloheptyl]methyl}pyrrolidin-2-one
(3aR,6aS)-1-oxo-5-[4-(1H-pyrazol-3-yl)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(pyridin-3-yl)-1-(3,4,7-trimethyl-1H-indole-2-carbonyl)piperidin-4-ol
8-(3-propyl-1H-pyrazole-4-carbonyl)-1-oxa-8-azaspiro[4.5]decane
N-[1-(5-propylpyrimidin-4-yl)piperidin-4-yl]-1-oxa-8-azaspiro[4.5]decan-3-amine
(3aR,6aS)-1-oxo-5-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)pyrazolo[1,5-a]pyridine-7-carboxamide
3-[({3-[3-(azepan-1-yl)-2-hydroxypropoxy]phenyl}methyl)(methyl)amino]propanamide
2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenyl)-6-(3-methylpyrazin-2-yl)-3,4-dihydropyrimidin-4-one
4-{pyrazolo[1,5-a]pyridine-7-carbonyl}-1,4-oxazepan-6-ol
5-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]pyridin-2-amine
1,3-dimethyl-4-{2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetyl}piperazin-2-one
4-[2-(trifluoromethyl)benzoyl]piperazine-2-carboxylic acid
(3S,4R)-1-(6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
4-[2-(2,4-dichlorophenyl)pyridine-4-carbonyl]morpholine
[(4-{2-[4-(3-chlorobenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(quinolin-6-ylmethyl)amine
1-{2-[1-(4-tert-butylbenzoyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
(1S,5R)-6-benzyl-3-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[3-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-4-(furan-2-ylmethyl)piperazine-1-carboxamide
7-(2-methoxyethyl)-2-(3-methylbutyl)-2,7-diazaspiro[4.5]decan-6-one
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
3-[2-(4-methoxyphenyl)ethyl]-5-methyl-5-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
2-cyclooctyl-4-(4-cyclopropanecarbonylpiperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
3-(1H-1,3-benzodiazol-1-yl)-N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]propanamide