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N-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
2-[4-methyl-6-({5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}amino)pyrimidin-2-yl]phenol
8-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
4-[1-(3-chlorophenyl)-1H-pyrazol-4-yl]-N-methyl-N-(pyrazin-2-ylmethyl)pyrimidin-2-amine
1-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(pyrrolidin-1-yl)ethan-1-one
4-(1H-imidazol-2-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine
2-[({1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}oxy)methyl]pyridine
ethyl 2-[(2-cyanophenyl)methyl]-2,7-diazaspiro[4.5]decane-7-carboxylate
3-chloro-N,6-dimethyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
3-(3-fluorophenyl)-4-{1H-imidazo[4,5-b]pyridin-2-yl}-1-(4-methoxyphenyl)-1H-pyrazole
2-methyl-N-{4-[(1-methylcyclohexyl)carbamoyl]phenyl}furan-3-carboxamide
6-fluoro-2-(1-methyl-1H-pyrazol-4-yl)-N-(propan-2-yl)-N-(pyridin-3-ylmethyl)quinoline-4-carboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(1H-pyrazol-1-yl)acetamide
N-(1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
2-[1-methyl-4-(3-methylbut-2-enoyl)-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl]acetic acid
2-(5-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridin-3-yl}-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-1-yl)ethan-1-ol
2-(3-hydroxypropyl)-9-(6-methyl-2-propylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-(4-methylphenyl)-5-[3-(propoxymethyl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-4-carboxamide
1-{1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]piperidin-4-yl}-3-methylbutan-1-ol
(1R,7S)-3-(2-ethoxyethyl)-N-methyl-4-oxo-N-(1H-pyrazol-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-{1-[(2,6-dimethoxyphenyl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N,1-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(2-ethyl-1H-imidazol-1-yl)-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]propan-1-one
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(3-fluoro-4-hydroxyphenyl)ethan-1-one
6-methyl-2-({4-phenyl-5-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-imidazol-1-yl}methyl)-3,4-dihydropyrimidin-4-one
N-{[1-(1,4-dithiepan-6-yl)piperidin-3-yl]methyl}-1H-indole-2-carboxamide
5-(3-methoxyphenoxymethyl)-N-(oxan-4-ylmethyl)-1H-pyrazole-3-carboxamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-(1,2-oxazolidin-2-ylmethyl)piperidin-2-one
2-{[(1-ethyl-1H-pyrazol-4-yl)methyl][(2-methylphenyl)methyl]amino}butan-1-ol
3-({1-[2-(2-hydroxyethoxy)ethyl]pyrrolidin-3-yl}methyl)benzamide
1-{3-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenyl}ethan-1-one
6-methoxy-2-oxo-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
(3S,4S)-4-(naphthalen-2-yl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-3-ol
2-(2-hydroxypropyl)-9-(3-methyl-1H-pyrazole-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[3-(morpholin-4-yl)propyl]amine
9-{2-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
3-(but-2-yn-1-yl)-5-(2-phenylethyl)-5-[1-(pyridin-4-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-3-(pyridin-4-yl)propanamide
1-(1H-imidazol-2-ylmethyl)-4-(2-methylphenoxy)piperidine-4-carboxylic acid
(2E)-N-{[3-methyl-7-(1H-pyrazole-4-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
5-chloro-4-{[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-2-methoxyphenol
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide
5-(oxolane-3-carbonyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(furan-2-ylmethyl)(1H-imidazol-2-ylmethyl)[2-(morpholin-4-yl)ethyl]amine
(1R,2R,6S,7S)-N-(2,3,5-trifluorophenyl)-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
11-[ethyl(2-methylprop-2-en-1-yl)amino]-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(3S)-3-benzyl-4-{[6-(dimethylamino)pyridin-3-yl]methyl}piperazin-2-one
2-methyl-8-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one