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2-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]-6-methylpyridine-3-carboxamide
3-[3-(3-fluoro-4-phenylbenzoyl)piperidine-1-carbonyl]pyridine
ethyl 1-[(4-methoxyphenyl)methyl]-5-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
ethyl 1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
2-methoxy-1-[1'-(pyridine-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
2-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-N-(1,3-thiazol-2-yl)propanamide
3-(1-methyl-1H-pyrazol-4-yl)-1-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
8-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-(4-chlorobenzoyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
5,6-dimethoxy-2-(4,4,4-trifluorobutyl)-1,2-dihydroisoquinolin-1-one
N-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]methyl}-2-(morpholin-4-yl)pyrimidine-5-carboxamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}oxane-4-carboxamide
1-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-phenylethan-1-one
ethyl 1-(2H-1,3-benzodioxole-5-carbonyl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
5-{[1-(2-methylphenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1,3,4-thiadiazol-2-amine
(2R,6S)-2,6-dimethyl-4-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}morpholine
N-cyclopropyl-1-{1-[(3,4-dimethylphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
N-[3-(2,6-dimethylphenoxy)propyl]-4-acetamido-N-methylbutanamide
(2S,4R)-N-ethyl-1-(furan-3-ylmethyl)-4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetamido]pyrrolidine-2-carboxamide
[3-({1-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-benzyl-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
N-benzyl-N-(2-hydroxyethyl)-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-ethyl-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-4-methyl-1,3-oxazole-5-carboxamide
5-(3-methyl-1,2,4-oxadiazol-5-yl)-2-[3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyridine
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-(5-methylpyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
9-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-6-oxa-9-azaspiro[4.5]decane
6-(cyclopropylamino)-N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]pyridine-3-carboxamide
(2S,4S)-N-ethyl-1-(1-ethylpiperidin-4-yl)-4-[2-(1H-imidazol-1-yl)acetamido]pyrrolidine-2-carboxamide
(3S,5S)-1-[(3-hydroxyphenyl)methyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxylic acid
1-(2-methoxyethyl)-8-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-hydroxy-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(4-methylphenyl)pyrimidine-5-carboxamide
3-methyl-N-(2-{2-[2-(pyrrolidin-1-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethyl)pyridin-2-amine
4-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-oxobutanamide
2-(2-{1-[2-(naphthalen-1-yl)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
(1S,4S)-3,3-dimethyl-2-methylidene-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]bicyclo[2.2.1]heptane-1-carboxamide
N-[(2,4-difluorophenyl)methyl]-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-5-phenyl-1H-pyrrole-2-carboxamide
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3-(3-methoxyphenoxy)azetidine
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-2-{4-[4-methyl-6-(methylamino)pyrimidin-2-yl]-1H-pyrazol-1-yl}acetamide
4-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-benzyl-3-methyl-8-({4-[methyl(phenyl)amino]phenyl}methyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-({1-[6-(cyclohexylamino)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
2-[3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanamido]-N-(4-fluoro-2-methylphenyl)propanamide
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(2,2-dimethyloxane-4-carbonyl)-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine