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N-{[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,3,5,7-tetramethyl-1H-indole-2-carboxamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[3-(pyridin-3-yloxy)propyl]benzamide
5-(azocane-1-carbonyl)-1-[2-(4-methoxyphenyl)ethyl]piperidin-2-one
N,N-diethyl-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine-3-carboxamide
N-benzyl-2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-sulfonamide
2-methyl-2-{4-[1-(1H-1,2,3,4-tetrazol-5-yl)-1H-pyrazol-4-yl]phenyl}propanenitrile
8-methoxy-2-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)quinoline
1-(5-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-ol
N-(2H-1,3-benzodioxol-5-yl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperidin-3-amine
(2S)-N-[3-(4-chlorophenyl)propyl]-1-(piperidin-4-yl)pyrrolidine-2-carboxamide
N-methyl-2-[3-oxo-1-({2-phenylimidazo[1,2-a]pyridin-3-yl}methyl)piperazin-2-yl]acetamide
7-methoxy-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-5-methylphenol
2-[1-(5-methanesulfonyl-2-methylpyrimidin-4-yl)piperidin-3-yl]-1,3-benzoxazole
4-ethyl-3-({1-[4-(methylsulfanyl)phenyl]-1H-1,2,4-triazol-5-yl}methyl)piperazin-2-one
(1S,2S)-2-{4-[2-(ethylamino)pyrimidine-5-carbonyl]piperazin-1-yl}cyclohexan-1-ol
9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-3-(thiophene-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-methyl-3-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[2-(1H-pyrazol-1-yl)ethyl]amine
2-(dimethylamino)-N-[2-methyl-5-({[1-(thiophen-3-yl)propan-2-yl]carbamoyl}amino)phenyl]acetamide
2-methyl-1-{6-methyl-5-[5-(3-methylfuran-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}propan-1-one
2-cyclopropanecarbonyl-8-(5-fluoro-2-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-[(4aR,7aS)-6,6-dioxo-4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
3-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-1-(1,2,3-thiadiazol-5-yl)urea
N-{[1-(dimethylamino)cyclohexyl]methyl}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
ethyl 1-(1-{2-[2-(3-fluorophenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carbonyl)piperidine-3-carboxylate
3-{[(1-{2-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-3-yl)oxy]methyl}pyridine
N-[(3-chlorophenyl)methyl]-N-methyl-2-oxo-1-phenylpyrrolidine-3-carboxamide
N-(3-phenylprop-2-yn-1-yl)-2-(propan-2-yloxy)-N-propylacetamide
N-{2-[2-(pyridin-2-yl)ethoxy]phenyl}morpholine-4-carboxamide
4-[1-(5-fluoro-2-methoxybenzoyl)azetidin-3-yl]pyridine
1-(dimethyl-1,3-thiazole-5-carbonyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
1-{3-[2-(4-methyl-1,4-diazepan-1-yl)-2-oxoethyl]morpholin-4-yl}-3-(pyridin-4-yl)propan-1-one
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-{[1-(pyridin-4-yl)propan-2-yl]amino}pyridine-3-carboxamide
2-benzyl-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-1,3-thiazole-4-carboxamide
1-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-5,5-diphenylpiperidin-2-one
3-chloro-N-(2-methoxyethyl)-4-{[1-(2-methylbutyl)piperidin-4-yl]oxy}benzamide
5-[4-(difluoromethoxy)phenyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-[7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-methoxyethan-1-one
[(5-fluoro-1H-indol-2-yl)methyl]({[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
3-({2-[5-(2-fluorophenyl)furan-2-yl]-1H-imidazol-1-yl}methyl)-5-(oxolan-2-yl)-1,2,4-oxadiazole
3-phenoxy-N-[1-({[1-(thiophen-2-yl)propan-2-yl]carbamoyl}methyl)-1H-pyrazol-4-yl]propanamide
N-ethyl-2-(furan-2-yl)-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-oxoacetamide
4-[(4-chloro-3-fluorophenyl)methyl]-3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
4-{2-[4-(propan-2-yloxy)phenoxy]ethyl}-1,3λ6,4-oxathiazinane-3,3-dione
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(3S,4S)-4-(4-fluorophenyl)-1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-3-ol
N-(2-fluoro-5-methylphenyl)-2-({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amino)acetamide
diethyl({3-[3-(morpholin-4-yl)azetidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine