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N-[1-(4-cyclopentylpyrimidin-2-yl)pyrrolidin-3-yl]-N-ethylacetamide
2-({[(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amino}methyl)benzoic acid
3-[2-(diphenylmethyl)-1H-imidazol-1-yl]propan-1-ol
4-(pyridin-3-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrimidin-2-amine
1-[3-(2-methylphenoxymethyl)piperidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1,3-thiazole-4-carboxamide
9-ethyl-4-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[(2-fluorophenyl)methyl]-N-[2-(1H-indol-1-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-methyl-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)propanamide
N-cyclopropyl-N-(1,3-thiazol-2-ylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
4-{[3-(2-{4-[2-(trifluoromethyl)benzenesulfonyl]piperazin-1-yl}ethoxy)phenyl]methyl}morpholine
6-[1-(adamantane-1-carbonyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
1-(propan-2-yl)-N-[1-(1,3-thiazol-2-yl)propyl]piperidine-4-carboxamide
(1S,5R)-6-[2-(methylsulfanyl)pyridine-3-carbonyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[3-({1-methyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}carbonyl)piperidin-1-yl]acetamide
(4aS,8aR)-6-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
5-chloro-2-methoxy-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
3-[4-(3-methylphenyl)piperazin-1-yl]-1-[3-(pyridin-2-yl)azetidin-1-yl]propan-1-one
N-(2,5-dimethyl-3-{[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-pyrrol-1-yl)acetamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}but-3-enamide
5-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]pyrrolidin-2-yl}-3-methyl-1,2-oxazole
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(5-{[cycloheptyl(pyridin-3-ylmethyl)amino]methyl}-2-ethoxyphenyl)methanol
N-[(1R,2R)-2-(dimethylamino)-2,3-dihydro-1H-inden-1-yl]-3-(1H-pyrazol-1-yl)benzamide
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
N-benzyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
2-(4-methoxyphenyl)-5-{[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyrimidine
1-[1-(hydroxymethyl)-9-[(4-methyl-1H-imidazol-5-yl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-(pyridin-4-yl)ethan-1-one
N-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-4-(pyridin-4-yl)piperidine-1-carboxamide
(1S,5R)-3-[(3-chloro-4,5-dimethoxyphenyl)methyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine
2-benzyl-4-(5-methoxyfuran-2-carbonyl)morpholine
7-(cyclobutylmethyl)-2-(4-methylquinolin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[3-(furan-2-yl)-3-phenylpropyl]-N-methyloxan-4-amine
2-{[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]methyl}benzoic acid
2-{[1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-yl]amino}-1-phenylethan-1-ol
1-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-{3-methylimidazo[1,5-a]pyridin-1-yl}-1H-1,2,3-triazole
3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-1-[3-(morpholin-4-ylmethyl)piperidin-1-yl]propan-1-one
1-{5-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-2-methylphenyl}imidazolidin-2-one
({4-[2-(1-cyclohexanecarbonylpiperidin-2-yl)ethoxy]phenyl}methyl)(methyl)(quinolin-5-ylmethyl)amine
methyl 2-{[2-(4-fluorophenyl)ethyl]sulfamoyl}-6-(2-methylpropanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
[(4-methanesulfonylmorpholin-2-yl)methyl]({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
4-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
3-methoxy-2-{[(oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}phenol
5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]quinoxaline
methyl (2S,3S)-2-{[5-(4-fluorophenyl)-1,2,4-triazin-3-yl]amino}-3-methylpentanoate
N-(butan-2-yl)-2-(phenylformamido)-N-(pyridin-4-ylmethyl)acetamide
1-cycloheptyl-5-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-2-one