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2-({[3-cyclopropyl-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)pyrimidine
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
5-(4-methanesulfonylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methylpiperidine
1-[(2-fluorophenyl)methyl]-4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-1,4-diazepane
N-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
1-[1-(hydroxymethyl)-9-(1H-imidazol-2-ylmethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-(pyrrolidin-1-yl)ethan-1-one
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[(4-methoxyphenyl)methyl]-3-{[(4-methyl-1H-imidazol-5-yl)methyl]amino}-5-(pyrrolidine-1-sulfonyl)benzamide
2-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-propoxyethan-1-one
2-[2-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
2-{[4-methyl-4-(methylsulfanyl)pentan-2-yl]amino}-N-(2-methylphenyl)acetamide
1-[(2-fluorophenyl)methyl]-6-oxo-N-{2-[4-(trifluoromethyl)phenyl]ethyl}piperidine-3-carboxamide
N-[(3-methoxyphenyl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-4-ethylcyclohexane-1-carboxamide
1-[4-({[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}amino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-methyl-5-(propan-2-yl)-N-[2-(pyridin-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
14-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]-6-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
3-{2-amino-4-methyl-6-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]pyrimidin-5-yl}propanoic acid
8-{[2-(methylsulfanyl)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[(4,6-dimethylpyridin-2-yl)methyl]-7-methoxy-N,4-dimethylquinazolin-2-amine
(2R,6R)-4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
(1H-imidazol-4-ylmethyl)(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
2-[(3,4-difluorophenyl)methyl]-8-(1-methylcyclopropanecarbonyl)-2,8-diazaspiro[4.5]decan-3-one
(2R,3S,6R)-3-(4-fluorophenyl)-5-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}pyridine-3-carboxamide
2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
2-(2-hydroxyethyl)-8-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
7-(cyclopropylmethyl)-2-[2-(1H-1,2,3-triazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
5-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]isoquinoline
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-2-methoxypyridine-3-carboxamide
8-(2-methoxypyridine-4-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
8-(2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[2-({ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-5-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
N-({1-[(3,4-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)-2-(pyridin-2-yl)acetamide
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]pyridin-2-amine
4-[1-(2-fluorophenyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]cyclohexan-1-ol
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N,N-diethyl-4-{[2-(1H-indol-3-yl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethan-1-one
2-[1'-(4-methoxybenzoyl)-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl]acetamide
3-(2-{[ethyl(methyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl)-4,5,6,7-tetrahydro-1-benzofuran-4-one
2-methyl-N-{[4-(trifluoromethyl)phenyl]methyl}imidazo[1,2-a]pyridine-6-carboxamide
4-{[3-(difluoromethoxy)phenyl]methyl}-1-[(3-methylphenyl)methyl]piperazin-2-one
(1S,5R)-6-[2-(methylsulfanyl)pyridine-3-carbonyl]-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
2-{[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine