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(3aS,6aR)-5-(1-benzofuran-2-ylmethyl)-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
{[(3R,4S)-1-(cyclobutylmethyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
(1S,5R)-3-cyclobutanecarbonyl-6-(2-methoxypyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
6-(2-chlorophenyl)-N-(1-hydroxypropan-2-yl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
5-chloro-2-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxy]pyridine
N-{1-[1-(carbamoylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
N-benzyl-N-methyl-3-{1-[2-(pyrimidin-2-ylsulfanyl)acetyl]piperidin-4-yl}propanamide
ethyl 5-[(1-carbamoylcyclopentyl)carbamoyl]-1H-imidazole-4-carboxylate
6-methyl-5-{2-oxo-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(3-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-oxopropyl)acetamide
N-(1-{7-[(4-fluoro-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
(2S,4R)-4-(benzylamino)-N-(2-methoxyethyl)-1-(propan-2-yl)pyrrolidine-2-carboxamide
3-(2,2-dimethyloxan-4-yl)-3-ethyl-1-{4-[(trifluoromethyl)sulfanyl]phenyl}urea
3-(diethylamino)-N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}propanamide
8-benzyl-3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(cyclohexylmethyl)-1-(furan-3-ylmethyl)-1,4-diazepan-5-one
N-(2,4-dimethylphenyl)-2-({[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)acetamide
4-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}pyridine
2-[methyl(5-{[methyl(quinoxalin-2-ylmethyl)amino]methyl}pyrimidin-2-yl)amino]acetic acid
N-[2-(dimethylamino)ethyl]-4-(4-methyl-1H-indazol-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(2Z)-3-(3-fluorophenyl)-N-[(1s,4s)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexyl]prop-2-enamide
{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
N-(1-{[5-(2-fluorophenyl)furan-2-yl]methyl}piperidin-4-yl)methanesulfonamide
N-cyclopropyl-4-[3-(2-ethylphenoxy)azetidin-1-yl]pyridine-2-carboxamide
2-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}-N-(thiophen-2-ylmethyl)quinazolin-4-amine
4-{2-[1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)piperidin-2-yl]ethyl}morpholine
methyl 9-[(4-fluorophenyl)methoxy]-3-{[4-(methoxycarbonyl)phenyl]methyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[(4-hydroxyadamantan-1-yl)methyl]-3H,4H-pyrido[4,3-d]pyrimidin-4-one
1-cyclohexyl-4-{3-[(4-ethylpiperazin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carbonyl}piperazine
1-(3,5-difluoropyridine-2-carbonyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
3-[4-(dimethyl-1,3-thiazole-4-carbonyl)piperazin-1-yl]-1-azabicyclo[2.2.2]octane
N-[1-(2,4-dimethoxyphenyl)ethyl]-N-methyl-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
1-{2-[4-(2,3-dihydro-1H-inden-2-yl)morpholin-2-yl]ethyl}-3-ethylurea
{1-[1-(4-chlorobenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}(phenyl)methanol
1-methyl-N-{3-[5-methyl-4-({[2-(methylsulfanyl)-1,3-thiazol-4-yl]formamido}methyl)-1,3-oxazol-2-yl]phenyl}piperidine-3-carboxamide
N-(1-cycloheptylpiperidin-3-yl)-3-(pyrazin-2-yl)propanamide
1-[(2,6-difluorophenyl)methyl]-N-methyl-N-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
(4aR,7aS)-1-methyl-4-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3-{4-[(dimethylamino)methyl]phenyl}phenyl)methanol
(3S,4R)-N,N-dimethyl-1-(3-methylthiophene-2-carbonyl)-4-propylpyrrolidin-3-amine
methyl 4-{4-[4-(1H-pyrazol-4-yl)butanoyl]piperazin-1-yl}benzoate
1-(3-{2-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]-1H-imidazol-1-yl}phenyl)imidazolidin-2-one
2-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1-(3-methylbutyl)piperazin-2-yl)ethan-1-ol
3-[1-(2-chloro-4-fluorobenzoyl)piperidin-3-yl]-N-cyclopropylpropanamide
4-[methyl(1H-pyrazol-3-ylmethyl)sulfamoyl]-N-(oxolan-3-yl)benzamide
N-{[1-(hydroxymethyl)cyclopentyl]methyl}-N-methylbut-3-enamide
(4S)-4-amino-5-{4-[4-(methoxycarbonyl)phenyl]piperazin-1-yl}-5-oxopentanoic acid
3-({[1-ethyl-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]methyl}(methyl)amino)-1λ6-thiolane-1,1-dione
8-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-1-ethyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(1H-pyrazol-5-yl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidine