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5-methyl-4-(4-methylpiperazin-1-yl)-N-[2-(methylsulfanyl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
1-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]butanamide
3-chloro-N-cyclopentyl-N-(3-phenylprop-2-yn-1-yl)pyridine-4-carboxamide
4-[6-(5-fluoro-2-methylphenyl)pyridazin-3-yl]thiomorpholine
4-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-5,6-dimethylpyrimidine
1-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-propylurea
1-(5-amino-4-chloro-1H-pyrazole-3-carbonyl)-N,4-dimethylpiperidine-4-carboxamide
8-[(2-aminopyridin-3-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]-1-phenylethan-1-ol
4-[4-(ethoxycarbonyl)-4-[(4-methoxyphenyl)methyl]piperidine-1-carbonyl]pyridin-1-ium-1-olate
2-{2-[3-(4-chlorophenyl)piperidin-1-yl]-2-oxoethyl}-5-(dimethylamino)-2,3-dihydropyridazin-3-one
(1R,5R)-3-(2-methyl-4-phenylpyridine-3-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
4-(6-methoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-2-(1H-pyrazol-4-yl)quinoline
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
2-{3-[2-(3-methoxyphenyl)azetidine-1-carbonyl]phenyl}-1H-imidazole
5-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-1,3-dimethylimidazolidine-2,4-dione
(2R)-2-amino-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4-methylpentanamide
2-(2,4-difluorophenoxy)-1-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
2-(2-ethoxyphenyl)-5-methyl-4-(1H-pyrazol-1-ylmethyl)-1,3-oxazole
6-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-9H-purine
5-(3-methylbutyl)-3-(oxan-4-yl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
N-(1-{1-[(4-chlorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-fluorobenzamide
N-[(3S,4R)-1-(3-chloro-4-fluorobenzoyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
3-(1H-imidazol-1-ylmethyl)-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidine
2-(1-{[1-(4-methylpyridine-3-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
1'-[2-(morpholin-2-yl)acetyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-(2-phenoxyethyl)piperidin-4-ol
N,1,3-trimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
3-{5-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-(4-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-1,3-benzoxazole
2-[1-(3,4-dihydro-2H-1-benzopyran-3-yl)piperidin-4-yl]-5-fluoro-1H-1,3-benzodiazole
N-[4-(4-{[1-(1,3-thiazol-5-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]benzenesulfonamide
2-cyclobutanecarbonyl-7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-6-one
(3aS,6aR)-5-(3-methylfuran-2-carbonyl)-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-({[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
[(2-ethoxyphenyl)methyl](ethyl){[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
N-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[5-({5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)thiophen-2-yl]ethan-1-one
1-[1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-yl]-3-phenylpropan-1-one
3-(2H-1,3-benzodioxol-5-yl)-5-(oxolan-2-yl)-1,2,4-oxadiazole
1-(4-fluorobenzoyl)-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-[3-(3-methoxyphenyl)phenyl]-N-(1,2-oxazol-3-ylmethyl)piperidin-4-amine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-[1,2,4]triazolo[4,3-a]pyridin-3-amine
1-[1-(2,6-difluoro-3-methylbenzoyl)piperidin-4-yl]-3-phenylpropan-1-ol
1-benzyl-3-(2-methoxyphenyl)-6-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one