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2-methoxy-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2-methylpropanamide
2,3,6-trimethyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)quinoline-4-carboxamide
{1-[2-(morpholin-4-yl)benzoyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
N-[(2-ethoxyphenyl)methyl]-N,3,5-trimethyl-1H-indole-2-carboxamide
N,N-dimethyl-6-[2-(methylsulfanyl)phenyl]pyridine-3-carboxamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-4-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
7-chloro-4-{2,8-diazaspiro[4.5]decane-3-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
(butan-2-yl)({[5-(1H-pyrazol-5-yl)furan-2-yl]methyl})(pyridin-4-ylmethyl)amine
2-{[(3,4-dichlorophenyl)methyl]amino}-N-(1,3-thiazol-2-yl)propanamide
(1S,5R)-6-cycloheptanecarbonyl-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-(2,3-difluoro-4-methylphenyl)-1-(1,4-dioxan-2-ylmethyl)-3-(oxan-4-yl)-1H-1,2,4-triazole
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methylpyridin-2-amine
3-[({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-N-methylpyridin-2-amine
N-(2-{5,6-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-2-yl}ethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
N-({1-[(6-methoxy-2H-chromen-3-yl)methyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
N-{[(3S,4S)-3-hydroxy-1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]methyl}-2-methylbenzamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(morpholin-4-yl)pyrimidine-5-carboxamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-5-ethyl-1,3-oxazole-4-carboxamide
1-(6-methyl-2-propylpyrimidin-4-yl)-N-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-4-amine
6-ethyl-1-methyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-[4-(3,4-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2,4,6-trimethoxyphenyl)methyl]piperidine
(2S,4R)-N-ethyl-4-[4-(4-methoxyphenyl)-4-oxobutanamido]-1-methylpyrrolidine-2-carboxamide
2-methyl-6-{1-[(3-methylquinoxalin-2-yl)methyl]piperidin-3-yl}pyrimidin-4-ol
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3,3-dimethylbutan-1-one
4'-[(4-methoxypyridin-2-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
methyl 3-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
7-methyl-8-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methoxy}quinoline
3-{3-[3-(3-fluoropyridin-4-yl)phenyl]-1H-pyrazol-1-yl}propan-1-ol
[4-(1H-indol-3-yl)butan-2-yl][(2-methyl-1,3-thiazol-4-yl)methyl]amine
N-{1-[(4-phenylphenyl)methyl]piperidin-4-yl}oxane-2-carboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-(ethylamino)-4-methyl-1,3-thiazole-5-carboxamide
N-{2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}-6-methoxy-1H-indazole
2-{2-[6-amino-5-cyano-4-(3-ethenylphenyl)pyridin-2-yl]phenoxy}acetamide
6-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-3,5-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
ethyl 1-(1-carbamoylpiperidine-3-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
N-tert-butyl-2-({3-chloro-6-methylpyrazolo[1,5-a]pyrimidin-2-yl}formamido)acetamide
2-[2-(morpholin-4-ylmethyl)phenyl]-1,3-thiazole-4-carboxamide
3-{imidazo[1,2-a]pyridin-2-yl}-N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]propanamide
9-(3-chloro-4-methoxybenzoyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
2-(dimethylamino)-N-methyl-2-(2-methylphenyl)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
(3R,4S)-4-cyclopropyl-1-[3-(3-methoxyphenyl)benzoyl]pyrrolidin-3-amine
1-methyl-3-[5-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]-1-(quinolin-3-ylmethyl)urea
N-{[1-(1,3-benzothiazol-2-ylmethyl)piperidin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
3-[(3R,4S)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
N-cyclopentyl-N-[(2,4-dimethoxyphenyl)methyl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetamide
methyl({[(1R,5S,6R)-3-(morpholine-4-carbonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}){[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
2-(1-benzyl-3-oxopiperazin-2-yl)-N-methyl-N-[(3-methylpyridin-2-yl)methyl]acetamide
1-(2,5-dimethylphenyl)-4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-3-phenyl-1H-pyrazole