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N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}thian-4-amine
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-1,3-oxazole-4-carboxamide
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(4-methoxyphenyl)acetamide
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(3-methoxyphenyl)-6-methyl-4-[4-(2-oxopyrrolidin-1-yl)benzoyl]piperazin-2-one
(2S,4S)-4-amino-1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N,N-diethylpyrrolidine-2-carboxamide
4-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methoxypyrimidin-2-amine
6-(2-aminoethyl)-N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-N,2-dimethylpyrimidin-4-amine
4-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-1-(1-methylpiperidin-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
methyl 3-(2-methoxyacetamido)-5-[(3-methylbutyl)amino]-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(2S,4S)-N-ethyl-4-[2-(pyridin-2-yl)acetamido]-1-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
3-(pyrazin-2-yl)-1-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propan-1-one
4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1-[(2S)-pyrrolidine-2-carbonyl]piperidine
2-(methylsulfanyl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)pyridine-3-carboxamide
4-methyl-2-{2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]ethyl}-6-(trifluoromethyl)pyrimidine
1,3-dimethyl-N-{2-[1-(propan-2-yl)piperidin-4-yl]ethyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-{2-[3-(pyridine-3-carbonyl)piperidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
3-[(3R,4S)-1-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(4aS,7aR)-1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(1-benzofuran-2-yl)-3-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-1,2,4-triazine
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-cyclopropyl-1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-[(1-methyl-1H-imidazol-2-yl)methyl]urea
4,6-dimethyl-3-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
9-(2-hydroxyacetyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-butyl-8-[3-(pyridin-3-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{1-[1-(2-aminoacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-methoxybenzamide
1-[3-cyclopropyl-5-(2-methyl-1-benzofuran-5-yl)-1H-1,2,4-triazol-1-yl]butan-2-ol
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(1,2-thiazole-5-carbonyl)pyrrolidin-3-yl]methanol
3-methyl-1-{1-[6-(1H-pyrrol-2-yl)pyridine-3-carbonyl]piperidin-3-yl}butan-1-one
1-ethyl-6-oxo-N-[(3-phenylphenyl)methyl]piperidine-3-carboxamide
2-methoxy-N-[(5-{[2-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]acetamide
2-[4-(2-methylpropyl)-1,4-diazepane-1-carbonyl]benzonitrile
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(quinoline-7-carbonyl)piperidin-3-yl]propan-1-ol
3-(dimethyl-1H-1,2,4-triazol-1-yl)-N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-methylpropanamide
3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-N-propylpiperidine-1-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-3-phenyl-1H-pyrazole-4-carboxamide
ethyl[(1-ethyl-1H-pyrazol-4-yl)methyl][(2-propylpyrimidin-5-yl)methyl]amine
3-[(2R)-1-hydroxybutan-2-yl]-1-(4-phenyl-1,2,3-thiadiazol-5-yl)urea
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-3-(1-methylpiperidin-3-yl)propanamide
[1-(4-amino-5-methylpyrimidin-2-yl)piperidin-4-yl](1-methyl-1H-imidazol-2-yl)methanol
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-6-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
1-[(3,5-difluorophenyl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
2-[1-(2,3-dihydro-1H-inden-2-yl)-5-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-1H-1,2,4-triazol-3-yl]acetamide
2-(furan-2-yl)-N-[2-methyl-5-(2-oxopyrrolidin-1-yl)phenyl]azepane-1-carboxamide
(1-methyl-5-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
(1R,5R)-N,N-dimethyl-6-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2,3-dimethoxy-N-{[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]methyl}benzamide
N-butyl-3-({[2-(2-chlorophenyl)ethyl]amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
N-cyclopropyl-2-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]pyridine-4-carboxamide
2-(4-methyl-1,4-diazepan-1-yl)-2-[2-(methylsulfanyl)phenyl]acetic acid