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1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-cyclopropyl-2-(2,6-dioxo-1,3-diazinan-1-yl)-N-[(4-ethoxyphenyl)methyl]acetamide
1-methyl-4-(5,6,7,8-tetrahydroquinoline-3-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
ethyl 1-(2H-1,3-benzodioxol-4-ylmethyl)-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
2-(pyridin-3-yl)-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]pyrimidin-4-ol
N-(1-methoxybutan-2-yl)-2-methyl-1-benzofuran-5-carboxamide
3-(hydroxymethyl)-1-({3-methoxy-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}methyl)piperidin-3-ol
14-(1H-imidazol-2-yl)-2,17-diazatetracyclo[9.8.0.03,8.013,18]nonadeca-1(19),3(8),4,6,11,13(18)-hexaen-16-one
1-[(4-chlorophenyl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
1-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-phenylpiperidine-4-carboxamide
5-fluoro-1-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazole
3-(3-aminopyrrolidine-1-carbonyl)-N-[2-(5-methylfuran-2-yl)ethyl]benzene-1-sulfonamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-1-methyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
methyl (2S,4R)-1-methyl-4-[2-(methylamino)benzamido]pyrrolidine-2-carboxylate
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-3-(1,2-oxazinan-2-yl)propanamide
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclobutanecarboxamide
1-(4-{3-oxa-9-azaspiro[5.5]undecan-9-yl}piperidin-1-yl)butan-1-one
N-{[5,8-dimethoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(furan-2-ylmethyl)propanamide
2-{4-[(4-methanesulfonylphenyl)methyl]piperazin-1-yl}-3-methylpyrazine
2-oxo-6-[(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)methyl]-1,2-dihydropyridine-3-carboxamide
4-(4-{[ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenyl)but-3-yn-1-ol
methyl 6-{[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]carbamoyl}pyridine-3-carboxylate
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
3-[4-(3-cyanopyrazin-2-yl)piperazin-1-yl]-N-(2-ethoxyphenyl)propanamide
1-[1-(2-cyclohexylacetyl)piperidin-3-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
5-{[(1,4-dioxan-2-ylmethyl)amino]methyl}-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-[1-(furan-2-ylmethyl)-4-(5-methylpyrimidin-2-yl)piperazin-2-yl]ethan-1-ol
(2,1,3-benzoxadiazol-5-ylmethyl)({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
3-(4-fluorophenyl)-1-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}pyrrolidine
6-ethoxy-2-[2-(4-methoxypiperidine-1-carbonyl)pyrrolidin-1-yl]-4-methylquinazoline
1-[1'-(3-hydroxypyridine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
5-(1-cyclohexanecarbonylpiperidin-4-yl)-5-[(4-fluorophenyl)methyl]-3-(oxolan-3-yl)imidazolidine-2,4-dione
1-[(4-chlorophenyl)methyl]-4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperazine
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(2-hydroxyphenoxy)ethan-1-one
3-[(3R,4S)-1-(1H-indole-6-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-(3,5-dimethyl-4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-pyrrol-2-yl)ethan-1-one
methyl N-(2-{2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)carbamate
N-[(2S,4R,6S)-2-benzyl-6-(2-fluoro-3-methoxyphenyl)oxan-4-yl]acetamide
4-propyl-1-(thiophen-2-ylmethyl)-1,4-diazepan-5-one
7-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-2-oxa-7-azaspiro[4.5]decane
N-methyl-5-{[methyl(2-phenylethyl)amino]methyl}-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide
2-amino-5-ethyl-4-[2-(ethylamino)pyrimidin-5-yl]-6-(propan-2-yl)pyridine-3-carbonitrile
4-[1-(1-ethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]benzoic acid
1-(2-methoxyphenyl)-4-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]piperazin-2-one
N-{2-[7-(2H-1,3-benzodioxol-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-4-methoxybenzamide
1-(2-ethoxyethyl)-N-methyl-2-oxo-N-[2-(pyridin-2-yl)ethyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-ethyl-4-[2-(pyridin-2-yl)pyrimidin-5-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-4,5,6-trimethylpyridine-3-carbonitrile
N,1-dimethyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1H-indole-2-carboxamide