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(3S)-N,N-dimethyl-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]azepan-3-amine
3-(piperazine-1-sulfonyl)-N-[2-(pyridin-4-yl)ethyl]benzamide
methyl 3-cyclobutaneamido-5-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]formamido}methyl)benzoate
[1-(5-fluoro-2-methylbenzenesulfonyl)-4-(2-phenylethyl)piperidin-4-yl]methanol
1-methyl-3-(2-methylpropyl)-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-pyrazole-5-carboxamide
2-[(3,4-dimethoxyphenyl)methyl]-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1,3-benzoxazole-6-carboxamide
1-(2-methoxyphenyl)-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1H-pyrazole-4-carboxamide
2-{[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]sulfonyl}benzonitrile
7-(2-methoxyethyl)-2-(2-methylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one
3-{1-oxaspiro[4.4]nonan-3-yl}-1-[3-(1,3-thiazol-4-yl)phenyl]urea
3-{[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-3-phenylpropan-1-ol
1-[(3-chlorophenyl)methyl]-5-(4-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazole
1-[(2-chlorophenyl)methyl]-4-[(1-methylpiperidin-4-yl)amino]pyrrolidin-2-one
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]propanamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-2-phenoxyacetamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-1-(pyridine-2-carbonyl)piperidin-4-amine
5-[3-(cyclohexylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-ethyl-3-methyl-1H-pyrazole
N-[(2-methylphenyl)methyl]-2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}acetamide
N-(1H-indol-5-yl)-4-(oxan-4-yl)piperazine-1-carboxamide
4-[1-(1-{1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}piperidin-4-yl)ethyl]morpholine
N-cyclopentyl-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,5-difluorobenzamide
3-{2-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}azepan-2-one
5-[(1,3-benzothiazol-2-ylmethyl)amino]-1-benzyl-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-[(2-fluorophenyl)methyl]-1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-1,4-diazepan-5-one
6-[methyl(2-methylpropyl)amino]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
methyl 2-[(cyclohexylmethyl)sulfamoyl]-6-(2-methylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-(3-chloro-4-methoxybenzoyl)-1-methylpiperazine-2-carboxylic acid
3-({[2-(1H-imidazol-2-yl)ethyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanamide
1-[2-({[(2-chlorophenyl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
(benzylsulfamoyl)[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]amine
2-{4-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]piperidin-1-yl}-7-methanesulfonyl-4-methylquinazoline
3-(8-methoxyquinolin-5-yl)-1,2-dihydropyridin-2-one
3-methyl-6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridazine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
N-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-[3-(2-methoxyphenyl)phenyl]-2,4-dimethyl-3-oxopiperazine-1-carboxamide
methyl[(3-methylpyridin-4-yl)methyl]{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}amine
{4-[(3-methoxyphenyl)methyl]-1-[1-(2-methoxyphenyl)propan-2-yl]piperidin-4-yl}methanol
3-{3-[3-(morpholin-4-yl)-3-oxopropyl]piperidine-1-carbonyl}-2H-chromen-2-one
[(3R,4R)-1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-2-[2-(trifluoromethyl)phenyl]ethan-1-one
1-({5-hexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
[(2S,6S)-4-(5-fluoro-2-methylbenzoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
4-[5-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoic acid
(2S)-2-amino-N-(2-{[(2-fluorophenyl)methyl]sulfanyl}phenyl)-3-(1H-imidazol-4-yl)propanamide
methyl 3-benzamido-5-{[(3,5-dimethoxyphenyl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[2-(3,4-dimethylphenoxy)acetyl]-1-(2-methylphenyl)piperazin-2-one
5-(naphthalen-2-ylmethyl)-5-{3-oxo-3-[3-(2-phenylacetyl)piperidin-1-yl]propyl}pyrrolidin-2-one