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2-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]benzamide
4-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methyl-6-propylpyrimidine
methyl 3-{4-[2-(2-chloro-6-fluorophenyl)acetyl]-2-oxo-6-(pyridin-4-ylmethoxy)-1,4-diazepan-1-yl}propanoate
[(1-{[1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]dimethylamine
2-({[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}amino)-N-(pyrazin-2-yl)acetamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(6-oxo-1,6-dihydropyridine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-({5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-yl}amino)propan-2-ol
methyl 3-(1,3-dimethyl-1H-pyrazole-5-amido)-5-{[2-(thiophen-2-yl)acetamido]methyl}benzoate
1-(4-{[1-(2-ethoxyethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}piperazin-1-yl)propan-1-one
(4aS,8aR)-6-(3,6-dimethylpyrazin-2-yl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-cyclopentyl-2-({[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}amino)propanamide
2-[1-(4-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-cyclobutylacetamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
methyl 9-[(4-fluorophenyl)methoxy]-3-{[4-(methylsulfanyl)phenyl]methyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}[(2-methyl-1H-imidazol-4-yl)methyl](oxolan-2-ylmethyl)amine
1-[(1-{[1-(3,6-dimethylpyrazin-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]piperidin-4-amine
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(propan-2-yl)amine
methyl 4-[2-(morpholin-4-yl)-2-(pyridin-3-yl)acetyl]piperazine-1-carboxylate
3-[(3S,4R)-1-(2-methylpropyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]-1-(pyrrolidin-1-yl)propan-1-one
1-{2-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]pyrimidin-4-yl}piperidin-3-ol
N-cyclobutyl-1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-amine
N-[3-(2-oxopyrrolidin-1-yl)propyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-(oxan-4-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
5-{[(benzylsulfamoyl)amino]methyl}-N-methylfuran-2-carboxamide
2-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1-methyl-1H-imidazole
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-3-(2-oxopyrrolidin-1-yl)benzamide
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}azepane
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}propanamide
1-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-4-(1H-pyrazol-1-yl)butan-1-one
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
N-cyclopentyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
(3S,4R)-4-(3-methoxyphenyl)-1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)pyrrolidine-3-carboxylic acid
7-(2-methoxyacetamido)-1-(2-phenylethyl)-N-[3-(pyridin-3-yl)propyl]-1H-1,3-benzodiazole-5-carboxamide
N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-(morpholin-4-yl)-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)propanamide
3-cyclopropyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1H-pyrazole-5-carboxamide
1-[4-(4-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
4-(8-methyl-3-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}imidazo[1,2-a]pyridine-2-carbonyl)morpholine
2-cyano-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)benzamide
5-[4-(4-methyl-1H-pyrazol-3-yl)piperidine-1-carbonyl]pyridin-2-amine
N4-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]pyrimidine-4,6-diamine
(3S,4S)-4-methyl-1-{[4-(2-methylpropyl)phenyl]methyl}piperidine-3,4-diol
1-[2-(1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
4-methyl-2-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}pyrimidine
5-[2-(ethylamino)ethyl]-1-(naphthalen-1-ylmethyl)pyrrolidin-2-one
(1S,5R)-6-(4-methylpyrimidine-5-carbonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(4aS,7aR)-1-(3-methyl-1H-pyrazole-5-carbonyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{5-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-4-phenyl-1H-imidazol-1-yl}propan-1-ol