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N-benzyl-5-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}pyrimidin-2-amine
6-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]quinoxaline
2-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidine
(2R,6R)-4-(1,1-dioxo-1λ6-thiane-4-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(benzylsulfamoyl)({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl})methylamine
N4-methyl-N4-(1,2-oxazol-3-ylmethyl)-7-(1,3-thiazol-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-[3-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}methyl)phenoxy]acetamide
(3aR,7aS)-2-[(5-methoxy-1,3,4-thiadiazol-2-yl)methyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
(5S)-5-{[benzyl({[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]methyl}pyrrolidin-2-one
ethyl 1-(dimethylsulfamoyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
(4aR,7aS)-1-(cyclopropylmethyl)-4-(4-hydroxy-3-methoxybenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3-methoxyphenyl)methyl]-2-[2,6,6-trimethyl-4-oxo-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
7-(3,6-dimethylpyrazin-2-yl)-4-(3-hydroxybenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(3S,4R)-1-(butane-1-sulfonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
1-{1'-[2-(2-methylphenoxy)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]-4-(piperidin-1-yl)butanamide
2,2-dimethyl-N-[2-(N-methylmethanesulfonamido)ethyl]-1-(thiophen-2-yl)cyclopropane-1-carboxamide
1-[7-(hydroxymethyl)-9-(5-methyl-1,2,4-oxadiazol-3-yl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-methoxyethan-1-one
methyl 1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine-4-carboxylate
1-(1-cyclopentylpiperidine-4-carbonyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine
9-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
4-[(3-{[3-(2,6-dimethylphenoxy)azetidin-1-yl]methyl}phenyl)methyl]morpholine
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-[(5-methylfuran-2-yl)methyl]piperazin-2-one
1-(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)propan-1-one
2-[2-(1H-pyrazol-1-yl)ethyl]-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidine
2-(1H-pyrazol-1-yl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)acetamide
4-(4-fluorophenyl)-1-{3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzoyl}-1,2,3,6-tetrahydropyridine
ethyl 2-(1-{4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanoyl}piperidin-2-yl)acetate
N-[2-(5-cyano-2-methyl-1H-indol-3-yl)ethyl]pyrimidine-5-carboxamide
N-{[5-(1H-imidazol-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-methoxyacetamide
2-(2-{[3-(3-chlorophenyl)pyrrolidin-1-yl]methyl}phenoxy)ethan-1-ol
1-[4-(2-methylpyrrolidin-1-yl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
4-hydroxy-4-(hydroxymethyl)-N-[2-(4-methoxyphenyl)phenyl]azepane-1-carboxamide
2-{2-[1-(3-acetamidobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
5-[2-(diethylamino)pyrimidin-4-yl]-2-ethoxybenzoic acid
8-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-chloro-N-cyclopentyl-4-[(1-{spiro[2.3]hexane-1-carbonyl}piperidin-4-yl)oxy]benzamide
5-[4-(diphenylmethyl)piperazin-1-yl]-1-ethyl-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-3-(1,2-oxazolidin-2-yl)propan-1-one
4-({2-[2-hydroxy-3-(4-hydroxypiperidin-1-yl)propoxy]-5-methoxyphenyl}methyl)piperazin-2-one
2-(dimethylamino)-N-(2-acetamidoethyl)-2-(4-fluorophenyl)acetamide
(3S,4S)-4-cyclopropyl-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]pyrrolidine-3-carboxylic acid
3-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)-6-ethoxy-1,2-dihydroquinolin-2-one
methyl (2S,4R)-4-[2-(2H-1,3-benzodioxol-5-yloxy)acetamido]-1-methylpyrrolidine-2-carboxylate
2-[1-(2,2-dimethylpropyl)-4-[(3,4,5-trimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-[3-(4-phenylbenzoyl)piperidin-1-yl]but-2-yn-1-one
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-1-{6-oxa-9-azaspiro[4.5]decan-9-yl}propan-1-one
2-amino-6-(3-methyl-1-propyl-1H-pyrazol-4-yl)-4-{[(1s,4s)-4-aminocyclohexyl]methyl}pyridine-3-carbonitrile
methyl 1-[(3R,5S)-1-[(3-methylthiophen-2-yl)methyl]-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
5-(2,6-difluorophenoxymethyl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]-1,2-oxazole-3-carboxamide