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5-[1-(3-chlorobenzoyl)piperidin-4-yl]-3-[(4-fluorophenyl)methyl]-5-methylimidazolidine-2,4-dione
(3R,4R)-N-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidine-1-carboxamide
6-chloro-2-methyl-4-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]quinoline
(1R,5R)-6-[(8-methoxy-2H-chromen-3-yl)methyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-methyl-6-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
2-[4-(5-cyclopropyl-1-{4-[2-(trifluoromethyl)phenyl]pyrimidin-2-yl}-1H-pyrazole-4-carbonyl)piperazin-1-yl]ethan-1-ol
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
6-[2-(3,4-dichlorophenyl)morpholin-4-yl]-9H-purin-2-amine
2-(dimethylamino)-2-(3-methylphenyl)-N-{3-[(1-methylpiperidin-4-yl)oxy]propyl}acetamide
4-cyclobutyl-6-methyl-2-[4-(pyrrolidin-1-yl)piperidin-1-yl]pyrimidine
N-(pyridin-2-ylmethyl)-4-[3-(pyrrolidin-1-yl)pyrazin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-methyl-2-(thiophen-2-ylformamido)propanamide
(2S,4R)-1-(5-acetylthiophene-3-carbonyl)-4-amino-N,N-diethylpyrrolidine-2-carboxamide
1-(2-fluoro-6-methoxybenzoyl)-4-[(2-fluorophenyl)methyl]piperidine
5-({4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-2-methylpyrimidine
4-{2-[(4-oxopiperidin-1-yl)methyl]phenyl}benzamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(oxolan-3-yl)sulfamoyl]benzamide
2-(1-methyl-1H-indol-3-yl)-1-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}ethan-1-one
methyl 1-[(3R,5S)-1-(2-ethylbutyl)-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
5-[(3S)-3-aminopiperidine-1-carbonyl]-2-(4-methylphenyl)pyrimidin-4-ol
1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-[5-(thiophen-2-yl)furan-2-yl]propan-1-one
2-methyl-6-{2-[(5-methylthiophen-2-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
(4aR,7aS)-1-acetyl-4-[2-(3-chlorophenoxy)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-[(2S)-pyrrolidine-2-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}pyridine-4-carboxamide
5-(3,4-dimethylphenoxymethyl)-N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
(4aR,8aS)-1-[2-(3-methoxyphenyl)ethyl]-6-[4-(1H-pyrazol-1-yl)benzoyl]-decahydro-1,6-naphthyridin-2-one
1-[3-oxo-3-(pyrrolidin-1-yl)propyl]-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S)-2-[(2-amino-5-ethyl-6-methylpyrimidin-4-yl)amino]-4-methylpentan-1-ol
(3S,9aR)-3-(2-methylpropyl)-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(5-methylfuran-2-yl)-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}benzamide
N-methyl-N-[2-(2-oxopiperidin-1-yl)ethyl]-2-(pyrrolidin-3-yl)benzamide
N-methyl-N-(1-methylpiperidin-4-yl)-3-[1-(pyridazine-4-carbonyl)piperidin-3-yl]propanamide
1-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid
2-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3,4-dimethoxypyridine
3-[2-(3,4-difluorophenyl)ethyl]-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidine
{1-[1-(5-chloro-2-methoxybenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanamine
2-[5-methyl-2-(propan-2-yl)phenoxy]-N-[(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)methyl]propanamide
methyl 5-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
9-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]benzoic acid
2-(2-methoxyethyl)-9-[3-(pyridin-2-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
5-{2-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
methyl 7-oxo-3-[4-(1H-pyrazol-1-yl)butan-2-yl]-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-ethanesulfonamido-1-methyl-2-phenyl-N-[1-(thiophen-2-yl)propan-2-yl]-1H-1,3-benzodiazole-7-carboxamide
3-[5-(4-chlorophenyl)-1H-pyrrol-2-yl]-1-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]propan-1-one
N-(adamantan-2-yl)-5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-[(3-methoxyphenyl)amino]butanamide
4-{1-[2-(4-chlorophenyl)ethyl]-6-oxopiperidine-3-carbonyl}-1-phenylpiperazin-2-one