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4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidine
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-2-phenyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
9-methoxy-10-(pyrrolidine-1-carbonyl)-3-[(2,4,5-trimethylphenyl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-[(4-chlorophenyl)methyl]piperazine
(4aS,8aS)-2-[4-(3-hydroxy-3-methylbutyl)benzoyl]-decahydroisoquinolin-4a-ol
3-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-3-methyl-1-[3-(methylsulfanyl)phenyl]urea
4-methyl-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-1,2,3,6-tetrahydropyridine
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl][(3-methoxyphenyl)methyl](prop-2-en-1-yl)amine
N-benzyl-N-methyl-3-(1-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanoyl}piperidin-4-yl)propanamide
1-tert-butyl-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
5-(2H-1,3-benzodioxol-5-yl)-N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-1,2,4-triazin-3-amine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-(2-methanesulfonylethyl)-1H-pyrazole-3-carboxamide
2-cyclopropanecarbonyl-8-[(5-ethylpyridin-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2-(2,5-dioxoimidazolidin-1-yl)acetamide
7-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-(methylsulfanyl)-1-[3-(phenylamino)piperidin-1-yl]propan-1-one
1-[1-(pyridin-2-ylmethyl)-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(1,3-thiazol-4-yl)ethan-1-one
1-(2-{1-[(4-methoxyphenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}piperidin-1-yl)ethan-1-one
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(4-methylbenzenesulfonyl)propan-1-one
N-(2-{5-[2-(dimethylamino)-1,3-thiazol-5-yl]-4-phenyl-1H-imidazol-1-yl}ethyl)-2-methylpropanamide
2-(4-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-(3-methylbutyl)piperazin-2-yl)ethan-1-ol
3-({[1-(hydroxymethyl)cyclopentyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
4-{4-[2-(dimethylamino)-2-(2-fluorophenyl)acetyl]piperazin-1-yl}benzonitrile
N-(2-hydroxyethyl)-1-methyl-3-(2-methylpropyl)-N-propyl-1H-pyrazole-5-carboxamide
1-(diphenylmethyl)-4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperazine
7-(1H-indazole-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-4-[2-(thiophen-3-yl)acetyl]-1,4-diazepan-2-one
N-cyclohexyl-3-{[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]amino}propanamide
N-(1-methylpiperidin-4-yl)-5-[1-(pyridin-2-ylmethyl)pyrrolidin-2-yl]thiophene-2-carboxamide
3-{5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenol
3-methyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-1H-pyrazole-4-carboxamide
2-{[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]methyl}-5-methoxyphenol
N-[3-(morpholin-4-yl)propyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-(4-{3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]propanoyl}piperazin-1-yl)benzoic acid
{1-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-2-(2-fluorophenyl)ethyl}[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
2-({3-[4-(3,4-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-3-methoxyphenol
2-(dimethylamino)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-2,3-dihydro-1H-indene-2-carboxamide
2-[6-(hydroxymethyl)-1,4-oxazepane-4-carbonyl]-4,6-bis(propan-2-yl)phenol
5-{[1-(morpholine-4-sulfonyl)pyrrolidin-3-yl]methyl}-1,2-dihydropyridin-2-one
8-[3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methylpropanoyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-cyclopentyl-1-(2-methylpropyl)-5-[3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
7-methyl-2-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
1-[(diethylcarbamoyl)methyl]-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[(3-methoxyphenyl)methyl]-4-(6-methylquinolin-4-yl)piperazin-2-one
N-{[3-(3-chlorophenyl)-1,2-oxazol-5-yl]methyl}-2-ethylpyrimidine-5-carboxamide
(1S,5R)-3-acetyl-N-(2-phenylphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(5-ethylpyridin-2-yl)methyl]benzamide
N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
3-{2-[5-(2,3-dimethoxyphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one