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1-(4-{[4-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
1-ethyl-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-(4-methoxybenzoyl)-4-(3-methyl-1,2-oxazole-5-carbonyl)piperazine
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-methyl-2-phenylpropan-1-one
4-(4-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperazin-1-yl)quinazoline
7-methoxy-3-(quinoxaline-2-carbonyl)-2,3,4,5-tetrahydro-1H-3-benzazepine
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)({[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl})amine
1-{[5-(2H-1,3-benzodioxol-5-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-3,3-dimethylurea
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
3-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
4-(5-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoic acid
ethyl[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
(2S,4S)-N-methyl-4-(4-{2-[(phenylcarbamoyl)amino]propan-2-yl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxamide
3,6-dimethyl-2-(1-propyl-1H-pyrazol-4-yl)-4-(pyrrolidine-1-carbonyl)quinoline
1-[2-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
2,6-dioxo-N-[(1-phenylpyrrolidin-3-yl)methyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(quinolin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2,2-dimethylpropyl 3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carboxylate
1-{2-[(1-benzofuran-2-ylmethyl)(methyl)amino]ethyl}cyclopentan-1-ol
1-[3-(4-phenylbenzoyl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
N,N-dimethyl-7-[4-(1H-pyrazol-1-yl)benzenesulfonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine
N-{[2-chloro-5-(trifluoromethyl)phenyl]methyl}-2-(1-methylpiperidin-4-yl)acetamide
2-[5-(1-cyclopropanecarbonylpiperidin-4-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]pyridine
2-cyclopropyl-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-1,3-benzoxazole-6-carboxamide
3-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1-(8-methylquinolin-5-yl)urea
[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl](methyl)(pyridin-2-ylmethyl)amine
1-[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-one
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
ethyl 1-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-3-(2-phenylethyl)piperidine-3-carboxylate
1-(4-methanesulfonylpiperazin-1-yl)-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
2-(1H-imidazol-4-yl)-1-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
methyl 3-{[1-(cyclopropylmethyl)-5-(2,4,5-trifluorobenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
2-methoxy-1-[3-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-carbonyl)piperidin-1-yl]ethan-1-one
1-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(thiophen-3-yl)ethan-1-one
2-methyl-4-{4-[4-(9H-purin-6-yl)piperazine-1-carbonyl]phenyl}butan-2-ol
2-({3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-1H-indole
N-{1-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]pyrrolidin-3-yl}acetamide
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-5-methyl-N-(thiophen-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
3-{1-[2-(propan-2-yloxy)propanoyl]piperidin-4-yl}benzonitrile
N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-2-methoxy-2-methylpropanamide
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
2-(methoxymethyl)-6-methyl-4-oxo-1-(3-phenylpropyl)-N-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
4-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-5,6,7,8-tetrahydroquinazolin-2-amine
2-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyrrolidine-1-carboxamide
N,N-dimethyl-2-[4-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)-1,4-diazepan-1-yl]acetamide
N-cyclopropyl-6-[4-(2-phenoxyethyl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
(3aS,6aS)-1-(3,4-difluorobenzenesulfonyl)-octahydropyrrolo[2,3-c]pyrrole
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-2-(methylamino)pyridine-4-carboxamide