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2-methoxyethyl N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)carbamate
(4aR,7aS)-1-(2-methylpropanoyl)-4-(2-phenylacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-acetyl-8-[2-(2,4-dimethylphenoxy)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-[4-(3-hydroxy-3-methylbutyl)benzoyl]-1-phenylpiperazin-2-one
[2-(1-benzyl-1H-pyrazol-4-yl)phenyl]methanol
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[(5-methylthiophen-2-yl)methyl]piperidine
2-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]pyridine-4-carbonitrile
2-{[(1R,5S,8R)-8-(dimethylamino)-3-azabicyclo[3.2.1]octan-3-yl]methyl}benzoic acid
1-[(2S,4R)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
(4aS,8aR)-6-(1,2-oxazole-3-carbonyl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2,2-dimethylpropyl 7-methyl-12-oxo-3,7,11-triazaspiro[5.6]dodecane-3-carboxylate
1-(3-acetylphenyl)-3-({1-[ethyl(methyl)amino]cyclopentyl}methyl)urea
2-[3-(propan-2-yl)-5-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]-1H-1,2,4-triazol-1-yl]pyridine
N-(1-{[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}piperidin-4-yl)methanesulfonamide
3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
1-methyl-4-{[5-(3,6,7-trimethyl-1-benzofuran-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidine
5-[(isoquinolin-5-ylmethyl)(methyl)amino]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
6-(2,6-dimethylquinoline-4-carbonyl)-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
5-{1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidin-4-yl}-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
2-[5-(ethylsulfanyl)thiophene-2-carbonyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
N-[3-(2-chlorophenoxy)propyl]-N-methyl-2-(2-oxoazepan-1-yl)acetamide
1-[3-(4-fluorophenoxy)propyl]-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperazine
5-oxo-1-(pyridin-3-ylmethyl)-N-[2-(1H-pyrrol-1-yl)ethyl]pyrrolidine-3-carboxamide
4-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}-3,5-dimethylphenol
2-(2-amino-2-methylpropanoyl)-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
2,4,5-trimethyl-6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
(2-{2-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
4-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
6-[4-(3-fluorophenoxy)piperidin-1-yl]pyridine-2-carboxylic acid
(4aS,8aS)-2-(4-chloro-2-methylbenzenesulfonyl)-decahydro-2,7-naphthyridin-4a-ol
2-{1-methyl-4-[2-(phenylamino)pyrimidine-5-carbonyl]piperazin-2-yl}ethan-1-ol
8-(1,3-benzothiazol-2-ylmethyl)-3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-(1H-indol-3-yl)ethan-1-one
1-ethyl-N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-5-oxopyrrolidine-3-carboxamide
5-{[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-N-ethylpyrimidin-2-amine
3-butyl-4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazole
2-[4-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)phenoxy]acetic acid
1,3-dimethyl-6-[4-(thian-4-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-4-(oxan-4-yl)piperazine
7-[(3,4-difluorophenyl)methyl]-2-(4-methyl-1H-imidazole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-cyclooctyl-2-{2-[(4-phenylpiperazin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}acetamide
[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)(quinolin-3-ylmethyl)amine
5-[1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
3-ethyl-1-(3-methylbutyl)-8-(3-phenylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-(cyclopropylmethyl)-2-(furan-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
3-methyl-5-(1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}pyrrolidin-2-yl)-1,2,4-oxadiazole
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]ethan-1-one
4-[(4-fluorophenyl)methyl]-1-methyl-3-(propan-2-yl)-1,4-diazepan-5-one
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidine-3-carboxylate
1-({5-[1-(2-aminopyrimidin-4-yl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol