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2-[(3-methoxyphenyl)methyl]-N-(thiophen-2-yl)morpholine-4-carboxamide
2-amino-4-(4-methoxy-3-methylphenyl)-6-(pyridin-2-yl)pyridine-3-carbonitrile
{3-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}[(4-phenylphenyl)methyl]amine
(4S)-4-amino-5-oxo-5-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}pentanoic acid
6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-(2-phenoxyethyl)piperidine-3-carboxamide
(2-methoxyethyl)({[3-(pyrimidin-2-yloxy)phenyl]methyl})(thiophen-2-ylmethyl)amine
4-(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)pyridine
2-(2-{[methyl({[3-(trifluoromethyl)phenyl]methyl})amino]methyl}phenoxy)acetic acid
(3S,4R)-3-methoxy-1-[(6-methylquinolin-5-yl)methyl]piperidin-4-amine
4-{[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]sulfonyl}-3-chlorobenzonitrile
N-[2-(1-hydroxycyclopentyl)ethyl]-6-methoxy-N,3-dimethyl-1-benzofuran-2-carboxamide
2-[(6-phenylpyridazin-3-yl)amino]-1-(pyridin-3-yl)ethan-1-ol
4-cyclopentyl-3-{2-oxo-2-[4-(pyridin-4-yl)piperazin-1-yl]ethyl}piperazin-2-one
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(pyrrolidin-1-yl)piperidine
2-{5-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
2-(2-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}phenoxy)acetic acid
N4-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N2,N2-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
2-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-N-(thiophen-2-ylmethyl)piperidine-3-carboxamide
1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(5-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
2-(2,5-dimethylphenyl)-2-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]acetic acid
2-amino-7-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[methyl(propan-2-yl)amino]-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
2-(2-butylpyrimidin-5-yl)-N-ethyl-N,3,6-trimethylquinoline-4-carboxamide
2-(hydroxymethyl)-N-[3-(methylsulfanyl)phenyl]azepane-1-carboxamide
3-(2-chlorophenyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-3-phenylpropanamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1-ethylpiperidine-2-carboxamide
1-[(2-methyl-1,3-thiazol-5-yl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
1-(4-methoxyphenyl)-3-methyl-5-(pyrrolidin-3-yl)-1H-1,2,4-triazole
[2-methoxy-1-(pyridin-2-yl)ethyl](methyl)[(3-methyl-1-benzofuran-2-yl)methyl]amine
1-{3-[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]phenyl}ethan-1-one
2-cyclopentyl-9-[(4-methoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-4-[(2-hydroxyethyl)sulfanyl]benzamide
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-propoxypropan-1-one
2-{1-cyclohexyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}pyridine
2-[1-(butan-2-yl)-3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-4'-yl]-N-ethylpropanamide
7-(2,6-dimethoxyphenyl)-9-methoxy-4-(pyridine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(dimethyl-1,2-oxazol-4-yl)-N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}acetamide
N-{2-oxo-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1,2,3,4-tetrahydroquinolin-7-yl}pyridine-3-carboxamide
N4-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}pyrimidine-4,6-diamine
1-[2-(4-fluorophenyl)piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
4-(8-methoxyquinolin-5-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
[(3S,5R)-1-(2-chloro-4-fluorobenzoyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
1-methyl-3-{[3-methyl-1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
2-[1-(2,2-dimethylpropyl)-4-(3-phenylprop-2-yn-1-yl)piperazin-2-yl]ethan-1-ol
2-(4-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperazin-1-yl)pyrimidine
(5S,9aS,9bS)-2-(2-phenylethyl)-5-[3-(1H-pyrazol-1-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-({4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)pyridine
5-{1-[2-(2,5-difluorophenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione