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2-(4-chloro-1H-pyrazol-1-yl)-1-[(3S,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
3-{2-oxo-2-[4-(thian-4-yl)piperazin-1-yl]ethyl}-2,3-dihydro-1H-isoindol-1-one
1-{1-[2-(2-chlorophenoxy)acetyl]piperidin-3-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
N-(1-benzothiophen-2-ylmethyl)-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamide
1-(2-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}phenyl)ethan-1-one
6-(1-cyclobutanecarbonylpiperidine-4-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine
3-{1-[1-(but-3-enoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea
(1R,7S)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-methyl-3-[(3-methylphenyl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[3-(dimethylamino)-2,2-dimethylpropyl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
1-[4-(2-fluorophenoxy)phenyl]-3-[3-(4-methylpiperazin-1-yl)propyl]urea
N-cyclopentyl-N'-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)butanediamide
3-(azocane-1-carbonyl)-N-(oxolan-3-yl)benzene-1-sulfonamide
4-{3-[4-(3-chlorophenyl)piperazin-1-yl]propyl}-1,4-oxazepan-6-ol
N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]cyclohex-3-ene-1-carboxamide
[(4-fluorophenyl)methyl]({imidazo[1,2-a]pyrimidin-6-ylmethyl})(oxolan-2-ylmethyl)amine
N-[(3S,4R)-3-benzyl-1-methylpiperidin-4-yl]-3-phenyl-1H-pyrazole-4-carboxamide
1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}piperidine-4-carboxamide
3-[(2S)-2-acetamidopropanamido]-N-(2-ethylphenyl)benzamide
[5-({[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})amino}methyl)furan-2-yl]methanol
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-1-[(2S)-4-methyl-2-(propan-2-yl)piperazin-1-yl]propan-1-one
1-{3,5-dimethyl-4-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1H-pyrrol-2-yl}ethan-1-one
(3S,4S)-1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
(3E)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-phenylbut-3-enamide
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
4-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-6-fluoro-1,3-benzothiazol-2-amine
4-({4-methyl-5-[1-(pyrrolidine-1-carbonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
7-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-methoxy-N-(pyridin-3-ylmethyl)acetamide
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
4-(4-{[4-(methylsulfanyl)phenyl]methyl}piperazin-1-yl)-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-(2-ethylpyrimidin-5-yl)-7-methyl-4-(pyrrolidine-1-carbonyl)quinoline
1-[2-({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]piperidin-3-ol
2-{5-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
(4-{5-[1-(1H-pyrazol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}phenyl)methanol
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-methyl-6-(2-methylpropyl)pyrimidine-4-carboxamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-(2-phenylethyl)-3-(propan-2-yl)-1H-1,2,4-triazole
1-cyclopentyl-3-(2-methylphenyl)-3-{2-oxo-2-[4-(pyridin-4-yl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
2-(1,2-benzoxazol-3-yl)-1-(1,2-oxazolidin-2-yl)ethan-1-one
1-cycloheptyl-5-{3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-2-one
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
3-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-N-(2-ethoxyethyl)benzene-1-sulfonamide
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2,2-dimethylpyrrolidin-3-amine
1-{2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]pyrimidin-4-yl}piperidin-3-ol
4-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1-ethylpyrrolidin-2-one
2-(dimethylamino)-N-methyl-6-(2-methylphenyl)-N-(2-phenylethyl)pyridine-3-carboxamide
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2-[4-(pyrrolidine-1-carbonyl)morpholin-3-yl]acetamide
1-(4-fluorophenyl)-4-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-3-yl}piperazine
N-[1-methyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
1-{imidazo[1,2-a]pyridine-6-carbonyl}-4-(2-methoxyphenoxy)piperidine
ethyl 1-(dimethylsulfamoyl)-4-(oxan-2-ylmethyl)piperidine-4-carboxylate