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N-[(3S,4R)-1-(3-methyl-1H-pyrazole-5-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
[(8-methyl-2-{octahydropyrrolo[1,2-a]piperazin-2-yl}quinolin-3-yl)methyl](thiophen-3-ylmethyl)amine
3-cyclohexyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-pyrazole-4-carboxamide
N-methyl-2-oxo-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
(1r,4r)-4-[({3-[2-hydroxy-3-(morpholin-4-yl)propoxy]phenyl}methyl)amino]cyclohexan-1-ol
3-{[(2,2-dimethyloxan-4-yl)amino]methyl}-1-(prop-2-en-1-yl)-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
{2-fluoro-5-[4-(morpholin-4-yl)phenyl]phenyl}methanol
2-{4-[(3,4-dimethoxyphenyl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[(5-chlorothiophen-2-yl)methyl]-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
methyl 3-[({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)[(3S)-2-oxoazepan-3-yl]sulfamoyl]thiophene-2-carboxylate
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-[3-(pyridine-2-carbonyl)piperidin-1-yl]ethan-1-one
2-[5-({2-[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}methyl)-1,2-oxazol-3-yl]pyridine
1-cycloheptyl-6-oxo-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}piperidine-3-carboxamide
propyl(pyridin-3-ylmethyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-cycloheptyl-6-oxo-N-(2-phenoxyethyl)piperidine-3-carboxamide
1-[4-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]amino}methyl)-2-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]methyl}piperidin-2-one
{3-ethyl-1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-3-yl}methanol
1-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-(2-cyclohexylethyl)-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-ethyl-N-(2-methylprop-2-en-1-yl)-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-[2-(methylsulfanyl)pyridine-3-carbonyl]-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
(3S,4S)-4-cyclopropyl-1-{[3-fluoro-2-(trifluoromethyl)phenyl]methyl}pyrrolidine-3-carboxylic acid
8-(propane-1-sulfonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[3-(4-methoxyphenyl)propyl]-6-(thiomorpholin-4-yl)pyridine-3-carboxamide
7-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-oxa-7-azaspiro[4.5]decan-8-one
2-(5-chlorothiophen-2-yl)-1-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-imidazole
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-4-(2,4-dioxoimidazolidin-1-yl)benzamide
N-[2-(4-chlorophenyl)ethyl]-2-{2-[(methylcarbamoyl)methyl]-3-oxopiperazin-1-yl}acetamide
N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-1-(propan-2-yl)piperidine-3-carboxamide
methyl 3-({[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}amino)propanoate
1-(4-chlorophenyl)-4-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine
ethyl 4-benzyl-1-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
7-[2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-[(2,4-dimethoxyphenyl)methyl]-5-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-3-yl}-4-methyl-1,3-thiazol-2-amine
(4aR,7aS)-1-cyclobutanecarbonyl-4-(4-ethylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}pyrimidine-5-carboxylic acid
(2S,4R)-4-amino-1-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[2-(2,4-dimethylphenoxy)ethyl]-N-methyl-4-(1H-pyrazol-4-yl)butanamide
3-{5-[2-(azocan-1-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
(1R,2R,6S,7S)-4-(2,4-dimethylquinoline-7-carbonyl)-4-azatricyclo[5.2.1.02,6]decane
(5S,9aS,9bS)-2-[(2-methylphenyl)methyl]-5-[3-(methylsulfanyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[4-({[3-(trifluoromethyl)phenyl]methyl}amino)piperidin-1-yl]pyridine-4-carbonitrile
N-ethyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-(2-methylprop-2-en-1-yl)acetamide
(2S,4S)-N-methyl-1-(naphthalen-1-ylmethyl)-4-{[(4-phenylphenyl)methyl]amino}pyrrolidine-2-carboxamide
[(1S,3R,3aS,6aR)-3-[(3Z)-hex-3-en-1-yl]-5-methyl-1-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-(pyrimidin-2-yl)-decahydroisoquinoline
methyl 9-[3-(dimethylamino)propoxy]-7-oxo-3-[4-(trifluoromethyl)benzoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}propanamide
8-(1,3-benzothiazol-2-yl)-1-(1H-imidazol-4-ylmethyl)-1,8-diazaspiro[4.5]decane