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8-chloro-2-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}quinoline
2-(1-{[1-(1H-indole-6-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
(3S,9aR)-3-benzyl-8-(naphthalene-1-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[(pyridin-2-ylmethyl)sulfamoyl]-5-(pyridin-3-yl)benzoic acid
1-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidin-1-yl)-2,2-dimethylpropan-1-one
3-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-1-[5-(dimethylamino)-2-methylphenyl]urea
4-{5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridine
3-[5-(2,1,3-benzoxadiazol-5-yl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
6-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-ylmethyl]naphthalen-2-ol
4-(2,2-difluoroethyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-({[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)amino}methyl)-4-hydroxyquinoline-6-carboxamide
2-ethyl-4-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
(3S,4S)-1-[3-(4-chlorophenyl)-1-phenyl-1H-pyrazole-4-carbonyl]piperidine-3,4-diol
2-cyclopropyl-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[3-(dimethylamino)pyrazin-2-yl]pyrrolidin-3-yl]methanol
2-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}benzoic acid
N-(1-{4-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)furan-3-carboxamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-1H-pyrazole-3-carboxamide
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
N-{[1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidin-3-yl]methyl}-1H-indole-2-carboxamide
1-benzyl-4-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-(1-methyl-1H-imidazol-2-yl)piperidine
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-5-chloro-3-methyl-1H-indole-2-carboxamide
(2S,4S)-N-ethyl-1-(furan-3-ylmethyl)-4-[3-(thiophen-2-yl)propanamido]pyrrolidine-2-carboxamide
methyl 5-[(4-hydroxybutan-2-yl)amino]-1-(2-methoxyethyl)-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-methyl-1-(2-{3-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoethyl)-1,4-dihydroquinolin-4-one
1-[6-(5-chlorothiophen-2-yl)pyridin-2-yl]piperazine
ethyl 3-[(4-fluorophenyl)methyl]-1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperidine-3-carboxylate
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
2-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N-(thiophen-2-ylmethyl)acetamide
N-(2-methoxy-5-methylphenyl)-2-{[6-(piperidin-4-yl)pyrimidin-4-yl]amino}acetamide
N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-3-(piperidin-3-yl)benzamide
1-(dimethyl-1,2-oxazole-4-carbonyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
3-(3-methoxyphenoxymethyl)-1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
1-ethyl-5-{[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(2R)-2-amino-1-[2-(2,5-dihydro-1H-pyrrol-1-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]-3-(ethylsulfanyl)propan-1-one
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-yl]propanamide
2-{methyl[4-(4-methylphenyl)-5-(quinolin-3-yl)pyrimidin-2-yl]amino}ethan-1-ol
3-(2,5-dimethoxyphenyl)-N-[4-(methylsulfanyl)phenyl]pyrrolidine-1-carboxamide
(4aS,8aR)-1-(3-hydroxypropyl)-6-(1,2-oxazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
4-fluoro-N-(2-{7-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
(3R,4R)-4-amino-1-{[2-(benzylamino)pyrimidin-5-yl]methyl}piperidin-3-ol
N-[(5-methyl-1H-pyrazol-3-yl)methyl]-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-cyclohexyl-N-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-ethyl-8-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(2-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}-2-oxoethyl)-3,4-dihydroquinazolin-4-one
5-acetyl-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]thiophene-3-carboxamide