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2-{4-[3-(methanesulfonylmethyl)piperidin-1-yl]-6-methylpyrimidin-2-yl}phenol
N-({1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-3-yl}methyl)-2-(2-methoxyphenoxy)acetamide
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-1-(pyrimidin-2-yl)piperidin-4-amine
2-(4-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}morpholin-2-yl)ethan-1-amine
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
4-(4-methyl-1,3-oxazole-5-carbonyl)-7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-phenyl-3-{1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}propanamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2,2-dimethylbutan-1-one
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-benzyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-1,2-oxazole-5-carboxamide
N,N-dimethyl-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3S,4S)-4-cyclopropyl-1-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]pyrrolidine-3-carboxylic acid
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[(3-methylthiophen-2-yl)methyl]-1H-pyrazole-3-carboxamide
3-methyl-5-[1-(pyrrolidin-1-yl)ethyl]-1-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
[(3R,4R)-1-[(5-ethylfuran-2-yl)methyl]-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
2-[(2-amino-6-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}pyrimidin-4-yl)amino]ethan-1-ol
N-(2-hydroxyethyl)-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N-methyl-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
methyl 3-[2-(2H-indazol-2-yl)acetyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(4-methylpyrimidin-2-yl)-4-(pyridin-3-yl)piperidin-4-ol
4-(3-{[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}propyl)piperazin-2-one
methyl 3-acetamido-5-[(4-methoxy-4-methylpentan-2-yl)amino]-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-methyl-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-chlorobenzamide
4-methyl-3-{1-[2-(2-phenylphenyl)-1H-imidazol-1-yl]ethyl}-4H-1,2,4-triazole
3-{[benzyl(3-hydroxy-2-methylpropyl)amino]methyl}benzonitrile
(3R,4S)-1-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)-4-propylpyrrolidin-3-amine
4-[2-chloro-5-(trifluoromethyl)benzoyl]piperazine-2-carboxylic acid
3-[1-(3-ethyl-4-methyl-1H-pyrazol-5-yl)-N-(2-phenylethyl)formamido]propanamide
1-[(3R,4R)-3-hydroxy-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-2-(2,3,6-trifluorophenyl)ethan-1-one
8-[1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
8-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-chloro-1H-pyrazol-1-yl)-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methylpropanamide
2-ethyl-4-{1-[4-(1H-pyrazol-5-yl)phenyl]-1H-imidazol-2-yl}pyrimidine
N-methyl-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-1-ethyl-1H-pyrazole-3-carboxamide
N-[(3S)-2-oxoazepan-3-yl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]-N-[3-(1H-imidazol-5-yl)phenyl]piperidine-1-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidine-2-carboxamide
2-cyclohexyl-5-{[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl}pyrimidine
1-[3-(1H-imidazol-1-yl)propyl]-2-(oxolan-3-yl)-1H-imidazole
1-cyclopentyl-4-[(4-methyl-1H-imidazol-5-yl)methyl]-1,4-diazepane
1-(2,3-dihydro-1H-inden-2-yl)-5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)pyrrolidin-2-one
N-({3-[2-(dimethylamino)ethoxy]phenyl}methyl)-3-methyl-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
4-(6-methoxyhexanoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
7-(cyclopropanesulfonyl)-N,N-dimethyl-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
8-{[3-(azocane-1-carbonyl)-1,2-oxazol-5-yl]methoxy}quinoline