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N-(3-ethylphenyl)-4-[2-(3-methoxyphenoxy)ethyl]piperazine-1-carboxamide
2-benzyl-8-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-2,8-diazaspiro[5.5]undecan-3-one
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
4-{[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
(1-{[(5-ethylpyrimidin-2-yl)(methyl)amino]methyl}cyclopentyl)methanol
(3aR,6aR)-2-(3-methylbenzenesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 4-{[(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-2-[(propan-2-yl)carbamoyl]pyrrolidin-1-yl]methyl}benzoate
(5S,9aS,9bS)-2-[(2-methylphenyl)methyl]-5-[3-(1H-pyrazol-1-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[4-(hydroxymethyl)piperidin-1-yl]pyridine-3-carboxamide
N-(1-{7-[(3-chlorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
methyl 3-(2,3-dimethylbenzamido)-6-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
[1-(dimethyl-1,3-thiazol-4-yl)ethyl]({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)cyclopropanamine
2-amino-4-(3-fluoro-4-hydroxy-5-methoxyphenyl)-6-(4-hydroxyphenyl)pyridine-3-carbonitrile
(2S,4R)-4-amino-1-(2,4-difluoro-3-methoxybenzoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[2-(3-fluorophenyl)ethyl]-4-{4-[(2S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
(4aS,7aR)-1-[(3-methylphenyl)methyl]-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[4-(2-phenylethyl)-1-{thieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl]methanol
N,N-dimethyl-2-[(2-phenoxypropanamido)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-2-(3-fluorophenyl)piperidine
N-methyl-3-(2-oxopyrrolidin-1-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]propanamide
1-cyclohexyl-4-[2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetyl]piperazin-2-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
4-(furan-2-carbonyl)-1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N-methyl-4-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1,3-thiazol-2-amine
4-methyl-N-(2-{7-[(2,3,4-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
1-[4-(1-acetylpiperidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
methyl 3-({[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}(oxolan-2-ylmethyl)sulfamoyl)thiophene-2-carboxylate
N,N-dimethyl-7-(3-methylfuran-2-carbonyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(1H-indol-3-yl)-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]ethan-1-one
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(furan-2-yl)azepane
1-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-5-methylphenyl)-1H-pyrazole
N-(2-methoxyethyl)-1-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
5-(3-chlorophenyl)-3-(2-hydroxyethyl)-6-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
3-(1-cyclohexyl-1H-pyrazol-5-yl)-1-(furan-2-ylmethyl)-1-(pyridin-2-ylmethyl)urea
{1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidin-4-yl}(thiophen-2-yl)methanol
5-(2-chlorophenyl)-2-methyl-N-(oxolan-2-ylmethyl)furan-3-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[(4-chlorophenyl)(pyridin-4-yl)methyl]acetamide
3-[(4-cyclopentylpiperazin-1-yl)methyl]-1-[(3,4-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
2-(phenylamino)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]pyrimidine-5-carboxamide
1-(7-{[3-(dimethylamino)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-methylpropan-1-one
7-[2-(2-methylphenyl)acetyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]acetamide
3-{[4-(4-fluorophenyl)-1,4-diazepan-1-yl]methyl}pyridin-2-amine
N-[4-(1H-pyrazol-1-yl)phenyl]-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-2-carboxamide
2-(2,3-dihydro-1H-inden-5-yloxy)-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-methylpropan-1-one
4-({4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
4-[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-pyrazol-4-yl]-1-(but-2-yn-1-yl)-1,2,3,6-tetrahydropyridine
2-(2-oxo-2-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}ethyl)-1,2-dihydrophthalazin-1-one
6-(aminomethyl)-N-[(1-ethylpyrrolidin-2-yl)methyl]-2-methylpyrimidin-4-amine