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4-[(2-fluorophenyl)methyl]-1-(2-methylbutanoyl)-1,4-diazepan-5-one
2-[(1-benzyl-1H-imidazol-2-yl)methyl]-5-(dimethylamino)-2,3-dihydropyridazin-3-one
4-hydroxy-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(thiophen-2-yl)pyrimidine-5-carboxamide
2-methyl-4-(5-{3-[4-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}furan-2-yl)but-3-yn-2-ol
N-cyclohexyl-4-[2-(phenylcarbamoyl)ethyl]piperidine-1-carboxamide
2-cyclopropyl-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]quinoline-4-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
N-(1-{1-[2-(2,4,6-trifluorophenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
3-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chloro-2-methylphenyl)urea
3-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
3-(furan-2-yl)-5-({2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}methyl)-1,2,4-oxadiazole
4-(3-fluorophenoxy)-1-(quinolin-5-ylmethyl)piperidine-4-carboxylic acid
7-(4-chlorobenzenesulfonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
(3aS,6aS)-2-[4-methoxy-3-(methoxymethyl)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(2-chlorophenyl)methyl]-4-ethyl-1,4-diazepan-5-one
2-[9-(3-methylpyrazin-2-yl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
N-(2-methoxyethyl)-2-(2-methoxyphenyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
1-(3-chlorophenyl)-5-methyl-4-[(3-methylquinoxalin-2-yl)methyl]piperazin-2-one
N-cyclopropyl-7-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-cyclopropyl-2-fluoro-6-hydroxy-N-[(2-methoxyphenyl)methyl]benzamide
N-[(3S,4R)-1-[2-(4-fluorophenoxy)ethyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
3-methoxy-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]propanamide
(1S,5R)-6-(2,6-dimethylpyrimidine-4-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
5-[(2-chlorophenyl)methyl]-3-(2-methoxyethyl)-5-[1-(2-methylpyridine-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[3-(1H-indol-2-yl)phenyl]-1-(1-methylcyclopropanecarbonyl)piperidine-3-carboxamide
N-(3,5-dimethoxyphenyl)-3-[1-(3,3,3-trifluoropropanoyl)piperidin-3-yl]propanamide
N-tert-butyl-3-oxo-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
(3R,4R)-1-{5-ethyl-6-methylthieno[2,3-d]pyrimidin-4-yl}-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
(1S,5R)-N-benzyl-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-(2-chloro-3,5-difluorophenyl)-3-methoxypyrrolidine-1-carboxamide
2-{4-[(4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazin-1-yl)methyl]phenoxy}acetic acid
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
N-(3-{[2-(2-aminoethyl)quinazolin-4-yl]amino}propyl)-4-methylbenzene-1-sulfonamide
2-(propan-2-yl)-4-[(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)methyl]pyrimidine
N-propyl-5-{[3-(pyridin-4-yl)azetidin-1-yl]methyl}pyrimidin-2-amine
N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)-4-(propan-2-yl)-1,2,3-thiadiazole-5-carboxamide
methyl 2-{[cyclohexyl(methyl)carbamoyl]methyl}-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
2-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}-N,N-dimethylbenzamide
N-methyl-N-(1,2-oxazol-5-ylmethyl)-2-(phenylamino)pyrimidine-5-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{3-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]piperidin-1-yl}acetamide
1-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
1-{6-[(1E)-pent-1-en-1-yl]pyridin-2-yl}piperazine
9-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
methyl 3-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]sulfonyl}thiophene-2-carboxylate
1-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-(methylsulfanyl)ethan-1-one
3-({[2-(furan-2-yl)ethyl]amino}methyl)-3-hydroxy-1-(2-phenylethyl)piperidin-2-one