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N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
N-ethyl-1-[(3-methoxyphenyl)methyl]-5-[2-(morpholin-4-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(dimethylamino)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-methyl-3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(oxolan-3-yl)propanamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[(1s,4s)-4-hydroxycyclohexanecarbonyl]pyrrolidin-3-yl]acetamide
N-[(4-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethoxy}-3-methoxyphenyl)methyl]-N-[(3S)-2-oxoazepan-3-yl]furan-2-carboxamide
8-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-phenyl-N-(1-{7-[(2,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
(1R,2R)-N-[2-(dimethylsulfamoyl)ethyl]-2-phenylcyclopropane-1-carboxamide
N-(1,3-benzoxazol-2-ylmethyl)-4-(3-hydroxy-3-methylbutyl)benzamide
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-3-(4-fluorophenyl)-1H-pyrazole-5-carboxamide
6-ethoxy-3-{[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-({7-[(3-phenoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenylacetamide
2-amino-4-ethyl-N-methyl-N-(quinolin-4-ylmethyl)-1,3-thiazole-5-carboxamide
2-{4-[(3,5-difluorophenyl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-methyl-N-[(3-methyl-1H-pyrazol-5-yl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
4-(3,6-dimethylpyrazin-2-yl)-N-[4-(1H-imidazol-1-yl)phenyl]piperazine-1-carboxamide
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-(4-methoxybenzoyl)-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperazine
2-[(5-hydroxy-6-methyl-1,2,4-triazin-3-yl)sulfanyl]-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}acetamide
N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-5-(piperidine-1-carbonyl)pyridin-2-amine
4-(1-ethyl-1H-pyrazole-4-carbonyl)-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
4-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
3-methyl-8-(2-methyl-4-phenylpyrimidine-5-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-(2-amino-6-methylpyrimidin-4-yl)-4-(3-phenylpropyl)piperidine-4-carboxylic acid
2-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidine-1-carbonyl]benzonitrile
5-(1-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-1H-imidazol-2-yl)-2-(methoxymethyl)pyrimidine
N-(2-fluorophenyl)-3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-cyclopentyl-4-{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}piperazine
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)[(1-methyl-1H-imidazol-2-yl)methyl](2-methylpropyl)amine
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(3,4-dimethylphenoxy)ethan-1-one
N-[(1S,3S)-3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}cyclopentyl]-1,2,5-thiadiazole-3-carboxamide
(3R,4R)-3-[ethyl({[4-methoxy-3-(methoxymethyl)phenyl]methyl})amino]-4-hydroxy-1λ6-thiolane-1,1-dione
2-(4-fluoro-3-methylphenyl)-2-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]acetic acid
1-(cyclopropylmethyl)-4-(3-methyl-1,2-oxazole-5-carbonyl)-2-(propan-2-yl)-1,4-diazepane
methyl 3-cyclohexaneamido-5-{[(1,3-dimethyl-1H-pyrazol-5-yl)formamido]methyl}benzoate
4-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-N-methylpyridin-2-amine
7-(1-benzothiophen-3-yl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{[(5-tert-butyl-1,3,4-oxadiazol-2-yl)amino]methyl}-6-ethyl-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-{[7-(2-phenylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine-2-carboxamide
N-(3,4-dimethoxyphenyl)-1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)piperidin-3-amine
6-chloro-1-methyl-N-{2-[methyl(phenyl)amino]propyl}-1H-indole-2-carboxamide
4-[1-(furan-3-carbonyl)piperidin-3-yl]-5-(4-methylphenyl)pyrimidine
1-[(2S)-2-hydroxy-2-phenylacetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-[(2R)-oxolan-2-yl]-3-(2-phenylethyl)-1,2,4-oxadiazole
5-fluoro-N4,N4-dimethyl-N2-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrimidine-2,4-diamine
1-[2-(1-methyl-1H-pyrazol-3-yl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one