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[4-(3,5,7-trimethyl-1H-indole-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
7-(3-methylbutyl)-3-(pyridin-4-yl)-2,4,5,7-tetraazatricyclo[6.4.0.02,6]dodeca-1(12),3,5,8,10-pentaene
1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-ol
3-(azocan-1-yl)-1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}propan-1-one
1-[(3S,5R)-3-(hydroxymethyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
N-[2-(pyridin-4-yl)ethyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methyl-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
N-[4-(pyridin-3-yloxy)phenyl]-1-(pyridin-4-ylmethyl)piperidine-4-carboxamide
1-(prop-2-en-1-yl)-5-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}ethan-1-one
2-[2-(1H-imidazol-4-yl)ethyl]-8-(5-methylpyrazine-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
4-oxo-5-phenoxy-1-[2-(pyridin-3-yloxy)propyl]-1,4-dihydropyridine-3-carboxylic acid
N-(2-methoxyethyl)-3-(1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-4-yl)propanamide
N-methyl-N-(oxolan-3-yl)-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
5-ethyl-5-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
9-hydroxy-3-[3-(phenylamino)piperidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
N-[(8-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]furan-2-carboxamide
N-(2-ethyl-1,3-dihydroxypropan-2-yl)-5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-5-propyl-1,2-oxazole-3-carboxamide
2-(4-chloro-1H-pyrazol-1-yl)-1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
1-{2-[({4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}methyl)amino]ethyl}imidazolidin-2-one
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine
4-(2-{1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-2-yl}ethyl)morpholine
N-methyl-N-(pyrazin-2-ylmethyl)-2-(pyridin-4-ylsulfanyl)acetamide
5-({3-[2-(3-chloro-4-fluorophenyl)pyridin-4-yl]pyrrolidin-1-yl}methyl)pyrimidine
3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-1-{imidazo[1,2-a]pyridine-3-carbonyl}piperidine
(2S,4S)-4-amino-1-[1-(methoxymethyl)cyclopropanecarbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]methylamine
2-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl)amino)propane-1,3-diol
2-(4-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-1-yl)acetic acid
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
1-cyclopropyl-5-oxo-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}pyrrolidine-3-carboxamide
5-fluoro-N4,N4-dimethyl-N2-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrimidine-2,4-diamine
5-ethyl-N4-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-6-methylpyrimidine-2,4-diamine
1-(4-methylphenyl)-3-{[1-(1-methylpiperidin-4-yl)piperidin-3-yl]methyl}urea
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-(phenylamino)pyrimidine-5-carboxamide
N-[(3S,4R)-4-(4-methylphenyl)-1-(1H-pyrrole-3-carbonyl)pyrrolidin-3-yl]cyclopropanecarboxamide
2-(azepan-1-yl)-N-{[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}acetamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-[3-(3-oxopiperazin-1-yl)propyl]acetamide
2-[3-(3-{furo[3,2-c]pyridin-4-yl}phenyl)-1H-pyrazol-1-yl]ethan-1-ol
N-(2-methanesulfonamidoethyl)-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
methyl 2-[1-(1H-indole-3-carbonyl)-3-oxopiperazin-2-yl]acetate
N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-1,2,3-triazole-5-carboxamide
N-[2-(benzyloxy)ethyl]-2-(pyrrolidin-3-yl)acetamide
(3aR,6aR)-2-cyclopropanecarbonyl-5-[(2-ethylphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2,3,4,9-tetrahydro-1H-carbazole-6-carboxamide
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-(2-methyloxolane-2-carbonyl)piperidine
5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1-methyl-1H-1,3-benzodiazole
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-phenylpiperidine