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5-(3,6-dimethyl-1-benzofuran-2-carbonyl)-2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(1H-indol-1-yl)ethan-1-one
2-hydroxy-1-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
1-(6-fluoro-4-methylquinazolin-2-yl)-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)pyrrolidine-2-carboxamide
(1S,5R)-3-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(5-chloro-2-methylphenyl)-3-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]urea
1-[(4-fluorophenyl)methyl]-4-[2-(1H-1,2,4-triazol-3-ylsulfanyl)acetyl]piperazin-2-one
3,6-dimethyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]pyrazin-2-amine
3-butyl-1-methyl-4-[1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carbonyl]piperazin-2-one
1-(4-{2-[(2-methylpyrimidin-4-yl)oxy]hex-5-en-1-yl}piperazin-1-yl)ethan-1-one
2-(4-phenoxybutanoyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
(4aR,6R,8aS)-2-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
N-ethyl-4-methyl-5-[3-(3-methylphenoxymethyl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
(2S,4R)-4-{4-[(2-cyclopentylacetamido)methyl]-1H-1,2,3-triazol-1-yl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
(4aR,7aS)-1-(2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}pyrimidin-4-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]-N-{[4-(trifluoromethoxy)phenyl]methyl}propanamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-[(1-hydroxycyclohexyl)methyl]acetamide
1-(4-fluorobenzenesulfonyl)-2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine
ethyl 2,4-dimethyl-5-{2-oxo-1-oxa-3,7-diazaspiro[4.5]decane-7-carbonyl}-1H-pyrrole-3-carboxylate
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N,6-dimethyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
methyl 3-benzamido-5-(cyclopentylamino)-1-(furan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[2-(dimethylamino)-6-methylpyrimidin-4-yl]-1,4-diazepan-2-one
{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}(methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
N-({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)cyclohexanecarboxamide
N-[2-(2-fluorophenyl)ethyl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
N-(3-chloro-4-fluorophenyl)-3-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}propanamide
1-(3-methylbutyl)-8-(2-methylpropyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(5-methylpyridin-2-yl)-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]piperidin-4-ol
1-({4-[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]phenyl}methyl)piperidine
N-{2-[5-(2-methyl-1,3-thiazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyridine-4-carboxamide
8-(but-3-enoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(1-cyclopropylethyl)-4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}benzamide
1-{1-[(3-chloro-5-ethoxy-4-hydroxyphenyl)methyl]piperidin-4-yl}piperidin-4-ol
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(quinolin-3-ylmethyl)propanamide
2-[methyl(phenyl)amino]-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
ethyl 2-[(5-{[2-(4-fluorophenyl)morpholin-4-yl]methyl}pyrimidin-2-yl)(methyl)amino]acetate
N-benzyl-N-methyl-2-[({[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amino)methyl]-2,3-dihydro-1H-inden-2-amine
(3S,4S)-1-[2-(4-fluorophenyl)ethyl]-4-methylpiperidine-3,4-diol
(2S,4R)-1-[2-(4-acetylphenoxy)acetyl]-4-amino-N-ethylpyrrolidine-2-carboxamide
N-[(2-chloro-4-fluorophenyl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-methyl-3-(2-phenylethyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-6-(piperidin-1-yl)pyrimidine
N,N-dimethyl-2-(pyridine-3-sulfonamidomethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-(4-ethoxy-3-methylphenyl)-4-{6-oxo-2,7-diazaspiro[4.5]decan-2-yl}butane-1,4-dione
4-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]acetyl}-1-[(3-fluorophenyl)methyl]piperazin-2-one
1-(carbamoylmethyl)-N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}piperidine-4-carboxamide
7-cyclobutaneamido-N-[2-(furan-2-yl)ethyl]-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
{1-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-2-phenylethyl}(2-methoxyethyl)(pyridin-2-ylmethyl)amine
6-{2-[1-(2-fluorophenyl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2,3-dihydropyridazin-3-one
7-(2-methoxyethoxy)-4-(3-methyl-1H-indol-2-yl)-1,2,3,4-tetrahydroquinolin-2-one