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N,N-dimethyl-6-(1,2,3,4-tetrahydroisoquinolin-5-yl)pyridine-3-carboxamide
ethyl 1-(3-methylbutyl)-5-(1-methylpiperidin-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2,5-dimethoxy-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
2-[5-(5-methyl-2-phenyl-1H-imidazol-4-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
1-(6-hydroxy-4-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
N-tert-butyl-2-[(1-hydroxypropan-2-yl)amino]acetamide
(1R,5R)-3-(4-chloro-3-fluorobenzoyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-methyl-2-[1-(1-methylpiperidin-4-yl)-4-phenyl-1H-imidazol-5-yl]-1H-1,3-benzodiazole
4-{1-[2-(oxolan-2-ylmethoxy)phenyl]-1H-imidazol-2-yl}pyridine
1-({4-methyl-5-[1-(pyridin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
3-[2-(2-fluorophenyl)ethyl]-1-[4-(propan-2-yl)-1,2,3-thiadiazole-5-carbonyl]piperidine
N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
methyl 4-(5-{[(3S,4S)-3-hydroxy-4-(pyrrolidin-1-yl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
N-[1-(4-fluorophenyl)ethyl]-N-methyl-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
2-[5-({2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-1H-pyrazol-3-yl]phenol
4-(4-methyl-1H-pyrazol-1-yl)-1-[3-(thiophen-3-yl)propanoyl]piperidine-4-carboxylic acid
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-[(3-methyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-({6-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]pyridin-3-yl}methyl)acetamide
3-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propyl]-1H-indole
1-(1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}azetidin-3-yl)-2-methylpiperidine
7-[(3-methylphenyl)methyl]-2-[2-(pyridin-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-methyl-5-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[4-(piperidine-1-carbonyl)piperidin-1-yl]propan-1-one
5-chloro-4,6-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-oxo-1,2-dihydropyridine-3-carboxamide
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)[(4-methyl-1H-imidazol-5-yl)methyl](oxolan-2-ylmethyl)amine
3-(3-fluoro-4-methoxybenzoyl)-1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidine
1-[(1-{6-[(1-methoxybutan-2-yl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
7-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
5-[1-(methoxymethyl)cyclopropyl]-1-(2-phenylethyl)-1H-1,2,4-triazole
(3S,4S)-1-{[3-chloro-5-methoxy-4-(prop-2-en-1-yloxy)phenyl]methyl}-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]propan-1-one
3-{1-[1-(5-methylhex-5-en-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
(4aR,7aS)-1-[(5-methylfuran-2-yl)methyl]-4-[2-(methylsulfanyl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(2-chlorophenyl)methyl]-N-(prop-2-en-1-yl)acetamide
1-({1-[6-(2-methylpyrrolidin-1-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
8-cyclopropyl-N-(2,4-difluorophenyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
5-(2,3-dimethoxyphenyl)-2-fluorobenzamide
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(furan-2-yl)-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
3-(1H-1,2,3-benzotriazol-1-yl)-1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]propan-1-one
1-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]-4-[(2-methylphenyl)sulfanyl]piperidine
N-cyclopropyl-1-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
7-(1H-1,3-benzodiazole-2-carbonyl)-2-methyl-2,7-diazaspiro[4.5]decane
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]({[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl})methylamine
1-ethyl-4,6-dimethyl-2-oxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,2-dihydropyridine-3-carboxamide
5-cyclopropyl-N-(1,4-dioxan-2-ylmethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-methyl-1H-pyrazole-4-carboxamide
5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
3-(3-chlorophenyl)-3-phenyl-N-[2-(pyrazin-2-yl)ethyl]propanamide
8-methanesulfonyl-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
4-(2-chloro-4-{[2-(dimethylamino)ethyl]carbamoyl}phenoxy)-N,N-dimethylpiperidine-1-carboxamide