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2-(dimethylamino)-2-(3-fluorophenyl)-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
4-(3,6-dimethylpyrazin-2-yl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperazine-1-carboxamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-chloro-3-methylbenzamide
4-(1-benzyl-1H-imidazol-2-yl)-1-(3-ethyl-1H-pyrazole-5-carbonyl)piperidine
N-[(3S,4R)-4-methoxyoxolan-3-yl]-4-[(pyridin-2-ylsulfanyl)methyl]benzamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-N,N-dimethyl-6-oxo-2,7-diazaspiro[4.5]decane-2-sulfonamide
6-[2-(benzyloxy)ethyl]-1,2-dihydroisoquinolin-1-one
4-(2,3-dihydro-1H-inden-2-yl)-3-{2-oxo-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethyl}piperazin-2-one
5-(4-benzoylpiperidine-1-carbonyl)-1-[(2-methoxyphenyl)methyl]piperidin-2-one
2-(dimethyl-1,3-thiazol-4-yl)-N-{1-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
4-(2-{[(4-fluorophenyl)methyl](methyl)amino}acetyl)-1-(4-methylphenyl)piperazin-2-one
5-(oxane-2-carbonyl)-N-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
[(2,2-dimethyl-1-phenylcyclopropyl)methyl]({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
N-[(5-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
4-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methoxypyrimidine
4'-(3,3-dimethylbutyl)-1-propanoyl-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(3aR,6aR)-2-(cyclobutylmethyl)-5-[2-(2-fluorophenyl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}-9-oxa-2-azaspiro[5.5]undecane
2-methoxy-5-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)benzoic acid
4-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2,4,5-trifluoro-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}benzamide
3-cyclohexyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-1H-pyrazole-4-carboxamide
14-(2-methoxy-4-methylphenyl)-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
1'-[2-(2-oxoazepan-1-yl)acetyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
4-[3-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,3-thiazole
1-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-3-(methoxymethyl)piperidine
N-[(2R,4R,6S)-2-cyclohexyl-6-(1-methyl-1H-imidazol-5-yl)oxan-4-yl]benzamide
6-(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)pyrimidin-4-ol
1-(3,5-dimethylphenyl)-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperazin-2-one
2-({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(2,2-dimethylpropyl)piperidin-3-yl]piperazine
1-(2H-1,3-benzodioxol-5-yl)-2-[5-(oxan-2-yl)furan-2-yl]-1H-imidazole
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
1-{2-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]phenyl}ethan-1-one
N-{[7-(2,3-dihydro-1-benzofuran-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2-phenoxyacetamide
4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-(1,2,3,4-tetrahydronaphthalen-2-yl)piperidine
6-[1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-3-yl]pyrimidin-4-ol
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-2-(pyridin-3-yl)acetamide
N-methyl-2-(methylsulfanyl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyridine-3-carboxamide
[(5-fluoro-1H-indol-2-yl)methyl]({[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl})methylamine
N-[(5-chloro-2-ethoxyphenyl)methyl]-N,1-dimethylpiperidine-2-carboxamide
1-benzyl-5-[butyl(methyl)amino]-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-1,3-thiazole-4-carboxamide
3-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-N,N-dimethylaniline
1-[(4aR,8aR)-7-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-(4-fluorophenyl)-1,4-diazepane
1-cyclopropanecarbonyl-N-[3-(1H-indol-2-yl)phenyl]piperidine-3-carboxamide
2-ethyl-8-(2-propoxybenzoyl)-2,8-diazaspiro[5.5]undecan-3-one