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5-(4-methylphenyl)-N-[(1R,2S)-2-phenylcyclopropyl]-1H-pyrazole-3-carboxamide
N-(oxolan-2-ylmethyl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-(pyridin-2-ylmethyl)propanamide
1-(4-{1-[(5-methylpyrazin-2-yl)methyl]-1H-1,2,3-triazol-4-yl}thiophen-2-yl)ethan-1-one
2-(4-{1-[2-(ethylsulfanyl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)ethan-1-ol
4-[3-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]piperazin-2-one
4-({1-[(2-fluoro-3-methoxyphenyl)methyl]piperidin-2-yl}methyl)morpholine
2-cyano-N-({1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)benzamide
2-{2-[bis(propan-2-yl)carbamoyl]phenyl}pyridine-4-carboxylic acid
4-{[methyl({[3-(methylsulfanyl)phenyl]methyl})amino]methyl}benzene-1,2-diol
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[6-(propan-2-yl)pyridin-2-yl]piperidin-3-yl]propanoic acid
1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-3-(1H-pyrazol-5-yl)piperidine
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-({1-[4-(1,3-thiazol-4-yl)phenyl]piperidin-4-yl}amino)butan-1-ol
3-[3-methyl-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]-4,5,6,7-tetrahydro-1H-indazole
3-cyclopropyl-5-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-1,2,4-triazole
N-cyclopropyl-2-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)acetamide
2-methoxy-2-phenyl-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N-methyl-4-{[(4-methylphenyl)amino]methyl}-N-(prop-2-yn-1-yl)benzamide
1-{2-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(pyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(2-chloro-5-fluorophenyl)-4-methoxy-4-(prop-2-en-1-yl)piperidine-1-carboxamide
N-[(2S)-1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-1-oxopropan-2-yl]acetamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyrazin-2-yl)ethyl]acetamide
6-methyl-4-[2-(trifluoromethyl)morpholin-4-yl]quinoline
N-cyclopentyl-2-({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)propanamide
4-methyl-2-phenyl-6-[3-(1H-pyrazol-5-yl)piperidin-1-yl]pyrimidine
3-hydroxy-1-(2-phenylethyl)-3-{[(propan-2-yl)amino]methyl}piperidin-2-one
1-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
2-[4-(4-chlorophenyl)butanamido]-3-(furan-2-yl)propanoic acid
(3S)-3-({[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)azepan-2-one
N-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-phenylbenzamide
2-[4-(aminomethyl)phenyl]benzamide
8-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-(4-ethylphenyl)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-cyclohexyl-4-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazine
5-methyl-4-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}-2-(thiophen-2-yl)-1,3-oxazole
3-(pentan-2-yl)-8-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-methyl-1-propyl-N-{3-[(pyridin-3-yl)amino]propyl}-1H-pyrazole-4-carboxamide
1-(5-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-1H-pyrazol-3-yl)ethan-1-one
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-(pyridazine-3-carbonyl)-1,4-diazepane
2-methyl-4-[3-(1H-pyrazol-3-yl)phenyl]pyrimidine
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methylacetamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-phenylprop-2-ynamide
1-[(3-fluorophenyl)methyl]-N-[(2-methylphenyl)methyl]-6-oxopiperidine-3-carboxamide
(3R,5S)-5-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyrrolidin-3-ol
4-[1-(pyrimidin-2-ylmethyl)piperidin-3-yl]benzoic acid
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]benzamide
1-(cyclohexylmethyl)-N-methyl-N-[4-(morpholin-4-yl)butyl]-1H-1,2,3-triazole-4-carboxamide
N-(1H-indazol-5-yl)-3-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)benzamide