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N-tert-butyl-3-(3-methanesulfonamidopropanamido)-2-methylbenzamide
(1S,5R)-6-[(4-fluorophenyl)methanesulfonyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-methyl-3-({[1-(2-phenylethyl)piperidin-4-yl]carbamoyl}amino)benzamide
3-cyano-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methylbenzamide
4-(dimethylamino)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
N-cyclopentyl-2-{[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]amino}propanamide
3-(3-chlorobenzoyl)-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
7-[(2,3-difluorophenyl)methyl]-2-(4-methyl-1,3-oxazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-(4-methyl-2-oxo-2H-chromen-7-yl)-2-(1,3-thiazol-2-yl)piperidine-1-carboxamide
3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}-N-(3-methoxyphenyl)piperidine-1-carboxamide
2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-4-carboxamide
(1R,5S,6R)-3-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
4-({4-[(4-ethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-3-ethylpiperazin-2-one
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[(5-methylthiophen-2-yl)methyl]pyrrolidin-3-yl]acetamide
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(1-phenoxypropan-2-yl)amine
4-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-2-(morpholin-4-ylmethyl)-1,4-oxazepane
[(4-{[1-(3-chlorobenzoyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(quinolin-6-ylmethyl)amine
5-chloro-N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-[4-(4-phenylpiperidine-1-carbonyl)piperidin-1-yl]-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
(1S,5R)-3-[(3,5-dichloropyridin-4-yl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(6-methylpyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-chloro-2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyrimidine
4-[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidin-1-yl]-2-[1-(thiophen-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-{[5-(2,4-dimethoxyphenyl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]methyl}pyridine
5-(6-aminopyridin-3-yl)-4-(4-methylphenyl)-N-(pyridin-3-ylmethyl)pyrimidin-2-amine
2-({[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)ethan-1-ol
methyl[2-(oxan-2-yl)ethyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
2-(2-methylphenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
1-(cyclopropylmethyl)-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-[(3-chlorophenyl)methyl]-N-(oxolan-2-ylmethyl)-1,3-benzoxazole-6-carboxamide
2,3-dimethyl-7-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}-1H-indole
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-[2-(5-methoxy-1H-indol-3-yl)ethyl]urea
[(2R)-1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}pyrrolidin-2-yl]methanol
2-[(oxolan-2-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(3aR,6aR)-2-(2-methoxyethyl)-5-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{[3-(4-methylphenoxymethyl)piperidin-1-yl]methyl}benzoic acid
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-3-[(4-methylphenyl)formamido]propanamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
2-amino-2-methyl-1-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]propan-1-one
5-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
(3S)-1-benzyl-N-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}pyrrolidin-3-amine
6-(4-methoxypiperidin-1-yl)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
N-[2-(pyridin-3-yl)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
{2-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}urea
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
2-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-1-(piperazin-1-yl)ethan-1-one
2-[(4-chlorophenyl)methyl]-N-methyl-N-[3-(morpholin-4-yl)propyl]-1,3-benzoxazole-5-carboxamide
2-[3-(1H-imidazol-1-yl)propyl]-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-oxo-2,3-dihydro-1H-isoindole-5-carboxamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-5-(morpholine-4-carbonyl)pyridin-2-amine
2-(6-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one