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N-(2-phenylethyl)-1-[1-(pyrimidin-2-yl)piperidin-4-yl]piperidine-3-carboxamide
4-[2-(2,3-difluorophenyl)acetyl]-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
N-benzyl-5-{[methyl(thian-4-yl)amino]methyl}pyrimidin-2-amine
(3S)-1-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-N,N-dimethylazepan-3-amine
5-(2-chlorophenyl)-N-[2-hydroxy-2-(pyridin-2-yl)ethyl]furan-2-carboxamide
1-cyclobutanecarbonyl-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
9-(1,4-dithiepan-6-yl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[2,5-dioxo-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
N-[2-(quinolin-6-yl)phenyl]cyclopropanecarboxamide
(2R,6R)-1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
1-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
N-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-2-fluoro-N-(oxolan-2-ylmethyl)benzamide
1-{4-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
2-{[(5-{[4-(furan-2-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl](methyl)amino}acetamide
(3R,4S)-1-[1-(3,4-difluorophenyl)piperidin-4-yl]-3,4-dimethylpiperidin-4-ol
6-chloro-2-[3-(1H-pyrazol-5-yl)piperidin-1-yl]quinoline
N-methyl-6-oxo-1-(2-phenylethyl)-N-(pyrazin-2-ylmethyl)piperidine-3-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(1-hydroxy-2-methylpropan-2-yl)benzamide
N-(2-hydroxyethyl)-5-{[methyl(2-phenylethyl)amino]methyl}-1,2-oxazole-3-carboxamide
(2E)-N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-5-methyl-N-(2-methylpropyl)thiophene-2-carboxamide
5-[4-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
3-(2-methylpropyl)-5-{[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2-oxazole
2-methoxy-1-[1'-(3-phenylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
3-fluoro-N-({7-[(3-phenoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
4,5,6-trimethyl-2-(3,4,5-trimethoxyphenyl)pyridine-3-carbonitrile
N-cyclopropyl-6-ethyl-N-(1H-indol-5-ylmethyl)-2-oxo-1,2-dihydropyridine-4-carboxamide
N-({1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-3-yl}methyl)-3,5-dimethoxybenzamide
2-[1-(3-methylpyrazin-2-yl)-1H-pyrazol-4-yl]ethan-1-ol
8-(4,6-dimethylpyridine-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-{[4-(2-chlorophenoxy)piperidin-1-yl]methyl}pyridin-2-amine
ethyl 4-[(4-methoxyphenyl)methyl]-1-[3-(prop-2-en-1-yloxy)benzoyl]piperidine-4-carboxylate
3-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-1,2-dihydroquinoxalin-2-one
3-({1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
4-methyl-5-{pyrazolo[1,5-a]pyridin-7-yl}-2-(4H-1,2,4-triazol-4-yl)pyridine
8-(5-acetylthiophene-2-carbonyl)-2-(oxolan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
N,2,3-trimethyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]quinoxaline-6-carboxamide
[3-(1H-imidazol-1-yl)propyl](pyridin-4-ylmethyl)(quinolin-2-ylmethyl)amine
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-amine
5-(2,6-difluorophenoxymethyl)-N-methyl-N-{[1-(2-methylpropyl)piperidin-4-yl]methyl}-1,2-oxazole-3-carboxamide
methyl 1-(3-{4-[(cyclohexylamino)methyl]phenoxy}-2-hydroxypropyl)piperidine-4-carboxylate
3-{5-[5-(oxolan-2-yl)thiophen-2-yl]-1,2,4-oxadiazol-3-yl}pyridazine
2-hydroxy-3-methyl-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}butan-1-one
1-[2-(methoxymethyl)piperidin-1-yl]-2-phenylethane-1,2-dione
N-{[7-fluoro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-1,3-thiazole-5-carboxamide
2-(1-{[1-(2,5-dimethylbenzoyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
3-(3,4-dimethoxyphenyl)-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
2-[2-(dimethylamino)ethyl]-9-(trimethyl-1H-pyrazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2-methoxyethyl)-7-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-[2-(diethylamino)ethyl]-N-methyl-1,2-oxazole-3-carboxamide