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4,4-difluoro-1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(methylsulfanyl)ethyl]acetamide
4-{1-benzyl-5-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperazin-2-one
6-[(3,4-dimethoxyphenyl)methyl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
1-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
4-(2-hydroxyacetyl)-1-(3-methoxyphenyl)piperazin-2-one
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl]methanol
2-[(6-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyrimidin-4-yl)amino]ethan-1-ol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)piperidin-3-ol
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-methyl-2-(morpholin-4-yl)propan-1-one
(4aS,7aR)-1-[(2-ethylpyrimidin-5-yl)methyl]-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-4-({methyl[(3-methylthiophen-2-yl)methyl]amino}methyl)benzene-1-sulfonamide
N-{3-[ethyl(phenyl)carbamoyl]phenyl}-2-methylpyridine-3-carboxamide
4-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(4-fluorophenyl)methyl]piperazin-2-one
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
(2S,4R)-N-ethyl-1-(thiophen-2-ylmethyl)-4-[2-(thiophen-3-yl)acetamido]pyrrolidine-2-carboxamide
N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
5-(2,6-difluorophenoxymethyl)-N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1,2-oxazole-3-carboxamide
1-(3-{[5-(3,4,5-trimethoxyphenyl)-1,2,4-triazin-3-yl]amino}propyl)pyrrolidin-2-one
N-(but-2-yn-1-yl)-3-[(2-fluorophenyl)formamido]-N-(furan-2-ylmethyl)propanamide
4-[2-(1-benzyl-3-oxopiperazin-2-yl)acetyl]-1-cyclopentylpiperazin-2-one
2-ethyl-8-[3-(furan-2-yl)-4-phenylbutanoyl]-2,8-diazaspiro[4.5]decan-3-one
3-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-3-methyl-1-(4-sulfamoylphenyl)urea
2-[2-chloro-4-(pyrrolidin-1-ylmethyl)phenoxy]-3-methoxypyrazine
2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2-oxo-1-phenylpyrrolidine-3-carboxamide
[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl](methyl){[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
N-[(3-methoxyphenyl)methyl]-3-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-yl)propanamide
1-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-2,2-dimethylpropan-1-one
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N,N-dimethylpyrimidine-5-carboxamide
1-methyl-N-[2-(2-methylpropanesulfonyl)ethyl]-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-cyclopentyl-1-[(4-methoxyphenyl)methyl]-5-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[(3R,4S)-1-{[4-(cyclopentyloxy)phenyl]methyl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1,3-dimethyl-N-[1-(pyridin-3-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}morpholine-2-carboxamide
5-{3-[(4-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-methyl-N-(1,2-oxazol-3-ylmethyl)pyridin-2-amine
3-(oxolan-3-yl)-5-(2,4,6-trimethylphenyl)-1,2,4-oxadiazole
methyl (2S,3S)-2-{[1-(cyclohexylmethyl)-5-(dimethylcarbamoyl)-4-oxo-1,4-dihydropyridin-3-yl]formamido}-3-methylpentanoate
(butan-2-yl)({[2-(methoxymethyl)pyrimidin-5-yl]methyl})(thiophen-3-ylmethyl)amine
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
1-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-(4-ethylpiperazin-1-yl)ethan-1-one
methyl({2-phenylimidazo[1,2-a]pyridin-3-yl}methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
8-[(1-methyl-1H-indol-3-yl)methyl]-3-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-methoxy-N-(1-{7-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
8-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[4-(adamantan-1-yl)piperazin-1-yl]-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
2-(4-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
1-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
3-(1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-1,3-oxazolidin-2-one