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(3S,4R)-1-(3,4-difluorobenzoyl)-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
4-{2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}-1-[(4-fluorophenyl)methyl]piperazin-2-one
2-{[(3aR,6aR)-2-methyl-octahydropyrrolo[3,4-c]pyrrol-3a-yl]formamido}-N-(2-methoxy-5-methylphenyl)acetamide
methyl 3-(furan-2-amido)-1-(3-methylbutyl)-5-[(2-methylbutyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(3,4-dimethoxybenzoyl)-1-(5-fluoro-2-methylbenzenesulfonyl)piperidine
1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-4-[(4-fluorophenyl)methyl]-1,4-diazepane
N-[1-(4-methanesulfonylphenyl)ethyl]-2-propylpyridine-4-carboxamide
(2S,4R)-4-amino-N-methyl-1-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}pyrrolidine-2-carboxamide
2-(6-methoxynaphthalen-2-yl)-4-(1-methyl-1H-pyrrole-2-carbonyl)morpholine
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
(1-{[(2-amino-6-ethyl-5-methylpyrimidin-4-yl)(methyl)amino]methyl}cyclopentyl)methanol
N-[1-(1H-imidazol-4-ylmethyl)azepan-4-yl]-3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[3-(piperidin-1-yl)propyl]acetamide
4-methyl-2-[1-(trimethylpyrimidin-4-yl)piperidin-4-yl]-1H-1,3-benzodiazole
8-[(4-methyl-1H-imidazol-5-yl)methyl]-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(2-methoxyphenyl)ethyl]-2,2-dimethyloxane-4-carboxamide
1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
1-(2-methyloxane-2-carbonyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
3-(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)phenol
methyl (2S)-2-{[1-cyclohexyl-5-(methylcarbamoyl)-4-oxo-1,4-dihydropyridin-3-yl]formamido}-2-phenylacetate
N-methyl-N-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}oxolan-3-amine
4-[(2-fluorophenyl)methyl]-3-{2-[4-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
5-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyridin-2-amine
4-(1-hydroxyethyl)-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
4-[5-(2-chlorophenyl)furan-2-carbonyl]-1-phenylpiperazin-2-one
{1-[2-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]piperidin-3-yl}methanol
5-[1-(2,2-dimethylpropyl)-4-hydroxypiperidin-4-yl]-N-[2-(3-fluorophenyl)ethyl]-1-benzofuran-2-carboxamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methylbut-2-enamide
2-[1-(cyclohexylmethyl)-4-[(2,3-dimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
[(5-methylthiophen-2-yl)methyl](oxolan-3-ylmethyl)(pyridin-4-ylmethyl)amine
N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
3-[(4-aminopiperidin-1-yl)sulfonyl]-N-(1,4-dioxan-2-ylmethyl)benzamide
1-(3-methoxyphenoxy)-3-{[5-(3-methoxyphenyl)-1,2,4-triazin-3-yl]amino}propan-2-ol
1-methyl-6-propyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-3-ol
1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-(propan-2-yl)piperazine
(2S,4R)-N,1-bis(propan-2-yl)-4-({[4-(propan-2-yl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
methyl({[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl})[1-(pyrimidin-4-yl)ethyl]amine
6-(3-{1-[2-(dimethylamino)ethyl]-1H-pyrazol-3-yl}phenyl)-N,N-dimethylpyrimidin-4-amine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
N-[(3R,4S)-1-(cyclobutylmethyl)-4-cyclopropylpyrrolidin-3-yl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetamide
4-(3-chlorobenzenesulfonyl)-7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(5-methyl-1,2-oxazol-3-yl)acetamide
(3S,4R)-1-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2-(methylsulfanyl)pyridine-3-carboxamide
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-(pyrimidin-2-yl)-1,4-diazepane
(1S,5R)-6-(3-ethyl-1H-pyrazole-5-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
4-[4-(3-methoxyphenyl)-5-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl]-1-[(5-methylthiophen-2-yl)methyl]piperidine
N5-[(1-ethyl-1H-imidazol-2-yl)methyl]-N5-methyl-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine