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N-(2-hydroxyethyl)-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]-N-(thiophen-2-ylmethyl)acetamide
4-cyclobutaneamido-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]benzamide
2-methoxy-3-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]pyrazine
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-({[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]amino}methyl)piperidin-2-one
ethyl 1-(thiophene-2-sulfonyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
(2S,4R)-1-cyclohexyl-N-[2-(2-methoxyphenyl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1-propylpiperidin-4-amine
N-(2-{4-[3-cyclopropyl-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]phenoxy}ethyl)acetamide
1-(2,3-dimethylquinoxalin-6-yl)-3-[2-(2-hydroxyethoxy)ethyl]urea
5-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazin-2-ol
1-{3-[(cyclohexylamino)methyl]phenoxy}-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
3-[2-oxo-4-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)piperazin-1-yl]benzonitrile
methyl 1-benzyl-3-(oxolane-2-amido)-5-(propylamino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)-1H-1,2,3-triazole-4-carboxamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
2-(5-acetylthiophen-3-yl)-N-[(2,3,6-trifluorophenyl)methyl]acetamide
1-tert-butyl-5-(2,3-dihydro-1-benzofuran-5-yl)-3-(oxan-4-yl)-1H-1,2,4-triazole
3-{1-[(3-methylthiophen-2-yl)sulfonyl]azetidin-3-yl}pyridine
ethyl(1H-imidazol-2-ylmethyl){[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
(1S,5R)-6-benzyl-3-(2,6-diaminopyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(furan-2-ylmethyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]piperidine-4-carboxamide
2-[3-methoxy-5-(trifluoromethyl)phenyl]-2-(thiomorpholin-4-yl)acetic acid
4-phenyl-N-({1-[3-(pyrazin-2-yl)propanoyl]piperidin-3-yl}methyl)benzamide
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
7-methyl-6-[2-(2-phenylethyl)morpholine-4-carbonyl]-1H,2H-pyrazolo[1,5-a]pyrimidin-2-one
N-[(2R,3R)-1'-[(4-chlorophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
1-cyclopentyl-6-oxo-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}piperidine-3-carboxamide
(1R,3S)-7-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-7-azaspiro[3.5]nonane-1,3-diol
1-[(2S)-4,4-difluoropyrrolidine-2-carbonyl]-4-[(3-fluorophenyl)methyl]piperazine
2-methoxy-N-{[5-(quinolin-5-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
1-(2-methoxyethyl)-6-oxo-N-[2-(propan-2-yloxy)ethyl]piperidine-3-carboxamide
1-(5-methyl-1,3,4-oxadiazol-2-yl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-(1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)propan-1-ol
6-[4-(4H-1,2,4-triazol-3-ylmethyl)piperazine-1-carbonyl]pyridin-2-amine
9-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
7-(4-propylpyrimidine-5-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-methoxy-5-{1-[3-(oxolan-3-yl)propyl]-4-phenyl-1H-imidazol-5-yl}pyrimidine
N-tert-butyl-2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
N-(1-{1-[4-(4-fluorophenyl)-4-oxobutanoyl]piperidin-4-yl}-2-(2-methylphenyl)ethyl)-N-methylcyclobutanecarboxamide
N-[2-(4-fluorophenyl)ethyl]-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
(dicyclopropylmethyl)(methyl){[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}amine
1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N,N-bis(prop-2-en-1-yl)piperidine-3-carboxamide
2-(furan-2-ylmethyl)-9-(oxolane-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(3-{2-methoxy-4-[(3-methylpiperidin-1-yl)methyl]phenoxy}propyl)-1,2,5-thiadiazole-3-carboxamide
(3R,5S)-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
1-methyl-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
1,3-dimethyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
8-[(2S)-2-amino-3-(1H-imidazol-4-yl)propanoyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{5-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]-1H-pyrazol-3-yl}phenol
({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)(methyl)[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amine