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N-[(4-methoxypyridin-2-yl)methyl]-4-(trifluoromethyl)pyrimidin-2-amine
N-{2-[7-(2,2-dimethylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-phenoxyacetamide
6-(4-hydroxyphenyl)-2-{3-[(3-hydroxypiperidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
3-(2-{2-[2-(4-chlorophenyl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethyl)-1,3-oxazinan-2-one
N-cyclopentyl-1-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
N-(1,3-benzoxazol-2-ylmethyl)-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-4-(4-methoxyphenyl)butan-1-one
[(2S,4R)-1-[6-(3-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-(dimethylamino)pyrrolidin-2-yl]methanol
1-(6-fluoro-4-methylquinazolin-2-yl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrrolidine-2-carboxamide
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
4-{[(isoquinolin-5-ylmethyl)(methyl)amino]methyl}benzonitrile
5-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]imidazolidine-2,4-dione
N-benzyl-5-{[3-(dimethylamino)-2,2-dimethylpropyl]amino}-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3,3-dimethyl-1-{2-oxo-2-[3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]ethyl}urea
[8-methyl-2-(3,4,5-trimethoxyphenyl)quinolin-3-yl]methanol
methyl 3-(cyclohex-3-en-1-ylmethyl)-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[(dipropylamino)methyl]-N-[(1-ethyl-1H-imidazol-2-yl)methyl]benzamide
N-[2-(4-fluorophenyl)ethyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-(pyridin-3-ylmethyl)acetamide
1-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}-3-(pyridin-4-yl)propan-1-one
[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl][(5-ethylpyridin-2-yl)methyl]methylamine
2-ethyl-9-(1,2-oxazole-3-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
2-[4-(6,7-dimethoxy-3-methyl-1-benzofuran-2-amido)-3,5-dimethyl-1H-pyrazol-1-yl]acetic acid
[(2S,4R)-4-(dimethylamino)-1-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}pyrrolidin-2-yl]methanol
N-(1H-indazol-6-yl)-7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
3-{[2-(1H-imidazol-4-yl)ethyl]sulfamoyl}-N-(oxolan-3-yl)benzamide
2-{2-[3-(1H-imidazol-1-yl)propyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-3-carboxamide
4-{[3-(2-hydroxyethyl)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl]methyl}-2,6-dimethoxyphenol
(2E)-3-(2-chlorophenyl)-N-cyclopropyl-N-({4-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]phenyl}methyl)prop-2-enamide
N-[1-(furan-2-yl)ethyl]-N-methyl-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
methyl 4-{[4-(3,5-dimethylphenyl)-3-oxopiperazin-1-yl]methyl}thiophene-2-carboxylate
3-[1-butyl-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-4-methoxybenzene-1-sulfonamide
4-{4-[(3,5-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}-2-methoxypyridine-3-carbonitrile
5-(1-ethyl-1H-pyrazol-3-yl)-4-phenyl-1H-imidazole
2-[5-(2,3-dihydro-1-benzothiophen-2-yl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
2-{4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-benzyl-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-acetamido-N,2-dimethyl-1H-1,3-benzodiazole-7-carboxamide
[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl][2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]methylamine
N-(1-{1-[2-(pyridin-3-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
2-(2-chlorophenyl)-N,3-dimethyl-N-propyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine
6-(2-chloro-6-fluoro-3-methylbenzoyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
6-[(3-hydroxy-3-methylpiperidin-1-yl)methyl]-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]acetamide
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
8-[(4-tert-butylphenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
1-(2-methoxyacetyl)-N-methyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidine-4-carboxamide
2-[(4aR,7aS)-6,6-dioxo-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
2-(pyridin-2-yl)-5-{[3-(pyrimidin-4-yl)piperidin-1-yl]methyl}pyrimidine
3-(1-methyl-1H-imidazol-2-yl)-6-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]pyridazine
1-[7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-pyrazol-1-yl)ethan-1-one