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(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-(2-phenylethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-methyl-3-(2-methylpropyl)-N-[2-(pyridin-3-yloxy)propyl]-1H-pyrazole-5-carboxamide
4-(2-propyl-1H-imidazol-1-yl)pyridine
3-[(cyclopropylmethyl)(2-methoxyethyl)carbamoyl]benzoic acid
2-(3-methylbutanoyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
6-[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]pyridine-2-carbonitrile
{3-[2-(1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]propyl}dimethylamine
[(5-{1-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1H-1,2,3-triazol-4-yl}thiophen-3-yl)methyl]dimethylamine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
1-(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzoyl)-4-(2-methoxyethoxy)piperidine
N-ethyl-1-methyl-N-[2-(2-methylphenoxy)ethyl]-4-oxo-1,4-dihydroquinoline-3-carboxamide
3-[(4-fluorophenyl)methyl]-5-methyl-5-[1-(5-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
3-[2-(4-fluorophenyl)ethyl]-1-(4-methyl-1H-pyrrole-2-carbonyl)piperidine
2-amino-4-(1H-imidazol-4-yl)-6-(2-methylbutan-2-yl)pyridine-3-carbonitrile
2-(2H-1,3-benzodioxol-5-yl)-2-[methyl(pyrazin-2-ylmethyl)amino]acetic acid
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-{[(3R,4R)-3-hydroxypiperidin-4-yl]amino}-6-(trifluoromethyl)pyridine-3-carboxamide
(1S,5R)-3-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-({1-[(3-methoxyphenyl)methyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
N-(2-methoxyethyl)-2-methyl-N-[(4-methylphenyl)methyl]imidazo[1,2-a]pyrimidine-3-carboxamide
N-[(2R,3R)-1'-[(5-chloro-2-hydroxyphenyl)methyl]-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
4-[(2-methylpyridin-3-yl)oxy]-1-[2-(pyrrolidin-1-yl)acetyl]piperidine-4-carboxylic acid
2-acetamido-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1,3-thiazole-5-carboxamide
1-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-4-yl)piperazine
1-[3-({3-[2-(methoxymethyl)piperidine-1-carbonyl]-1H-pyrazol-5-yl}methoxy)phenyl]ethan-1-one
6-[2-fluoro-6-(propan-2-yloxy)phenyl]pyridine-2-carbonitrile
N-cyclohexyl-5-{1-[(isoquinolin-5-ylmethyl)amino]ethyl}-N,4-dimethylpyrimidin-2-amine
2-(2-cyclopropylacetyl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
6-(2-chlorophenyl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
8-(1-benzofuran-2-ylmethyl)-1-ethyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[1-(3,6-dimethylpyrazin-2-yl)piperidin-4-yl]piperidin-3-ol
dimethyl({5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]furan-2-yl}methyl)amine
4-(1-methyl-1H-pyrazol-4-yl)-2-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]pyrimidine
4-(2-methyl-1-phenyl-1H-1,3-benzodiazole-5-carbonyl)piperazin-2-one
1-cyclopropyl-4-{[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-1H-imidazol-1-yl]methyl}pyrrolidin-2-one
8-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)butan-1-one
1-[1-(carbamoylmethyl)piperidine-4-amido]-1,2,3,4-tetrahydronaphthalene-1-carboxylic acid
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(3,4,5-trimethoxyphenyl)acetamide
9-(cyclopropanesulfonyl)-2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecane
2-{5-[4-(ethylamino)pyrimidin-2-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
5-{1-[2-(3-chlorophenyl)acetyl]piperidin-4-yl}-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
2-(5,6-dimethoxy-1-oxo-1,2-dihydroisoquinolin-2-yl)-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
4-fluoro-N-(2-{[(3-hydroxypiperidin-3-yl)methyl]amino}ethyl)benzamide
N-{[3-(2-methoxyethoxy)phenyl]methyl}-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[2-(cyclohexylmethyl)morpholine-4-carbonyl]pyridin-3-ol
N-methyl-N-(1-methylpiperidin-4-yl)-3-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)propanamide
5-[1-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-3-yl]-N-[(2,5-dimethoxyphenyl)methyl]-4-methyl-1,3-thiazol-2-amine
2-[4-(piperazin-1-ylmethyl)phenyl]-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one