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N-{2-[(5-ethyl-1,2-oxazol-3-yl)formamido]ethyl}pyridine-3-carboxamide
3-{[bis(propan-2-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-cyclopropyl-N-{[7-fluoro-2-(4-methoxyphenyl)quinolin-3-yl]methyl}-2-(thiophen-3-yl)acetamide
3-({1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)-2,3-dihydro-1,3-benzoxazol-2-one
6-{methyl[2-(morpholin-4-yl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
1-(3-carbamoylpyridin-2-yl)-4-(4-chlorophenoxy)piperidine-4-carboxylic acid
N-cyclohexyl-2-{1-[2-(dimethylamino)ethyl]-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl}-N-methylacetamide
N-methyl-N-[2-(2-oxopiperidin-1-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
2-(3-acetyl-1H-indol-1-yl)-N-[(1-ethyl-1H-imidazol-5-yl)methyl]butanamide
4-({5-[1-(2-ethyl-6-methylpyrimidin-4-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
3-{2-[5-(2,1,3-benzoxadiazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,3-oxazinan-2-one
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1,2-oxazolidin-2-yl)propanamide
{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyridin-2-yl)propan-2-yl]amine
(1S,3R)-3-amino-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}cyclopentane-1-carboxamide
1-[2-(methylsulfanyl)pyrimidin-4-yl]-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]piperidin-4-amine
[(3-fluorophenyl)methyl]({[6-(pyrrolidin-1-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})amine
4-methoxy-N-[2-({5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)ethyl]benzene-1-sulfonamide
3,5-dimethyl-N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}-1,2-oxazole-4-sulfonamide
2-[1-(2,2-dimethylpropyl)-4-(quinolin-6-ylmethyl)piperazin-2-yl]ethan-1-ol
{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}(1,2-oxazol-3-ylmethyl)amine
N-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
5-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]propanamide
(1S,4R)-2-{2-[1-tert-butyl-3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2-azabicyclo[2.2.1]heptane
(4aR,8aR)-2-cyclobutanecarbonyl-7-[(2-methoxypyridin-3-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
4-[4-(2-methylpropyl)-1,4-diazepan-1-yl]-4-oxobutane-1-sulfonamide
N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-1-benzothiophene-5-carboxamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-N-[3-(methylsulfanyl)phenyl]piperidine-1-carboxamide
(1S,5R)-3-benzyl-6-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
1-(pyridine-3-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
(4aS,8aR)-6-(4-methylpyrimidin-2-yl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-{6-[3-(2-chlorophenyl)pyrrolidin-1-yl]pyridin-3-yl}ethan-1-one
1-[3-(2-methoxyphenoxy)propyl]imidazolidin-2-one
N-[2-(2-methyl-1-phenyl-1H-indol-3-yl)ethyl]-2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)acetamide
N,2-dimethyl-6-(piperidin-3-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-4-amine
2-(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}pent-4-en-1-one
3-[(4-hydroxy-4-phenylpiperidin-1-yl)methyl]-7-methoxy-1,2-dihydroquinolin-2-one
1-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-4-(furan-2-carbonyl)piperazine
7-(cyclopropylmethyl)-2-(2-methyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-2-one
2-benzyl-N-(4-butylphenyl)-3-oxopiperazine-1-carboxamide
(4aS,7aR)-1-(2,5-dimethoxybenzoyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[5-({2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
4-ethyl-3-[1-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{[(3-methylthiophen-2-yl)methyl]amino}-N-(4H-1,2,4-triazol-4-yl)benzamide
2-methoxy-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
(3R,4R)-3-cyclopropyl-4-methyl-1-[3-(trifluoromethyl)benzoyl]pyrrolidin-3-ol
(3S,5S)-5-[1-(2,3-dihydro-1H-inden-5-yl)-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-1-methylpyrrolidin-3-amine