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N-(3-methanesulfonamidophenyl)-4-(4-methylphenyl)piperazine-1-carboxamide
1-benzoyl-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-amine
1-(carbamoylmethyl)-N-[cyclopropyl(6-methylpyridin-2-yl)methyl]piperidine-4-carboxamide
4-methyl-N-[2-(pyridin-2-ylmethoxy)phenyl]-1,4-diazepane-1-carboxamide
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-2-(pyrrolidin-1-yl)acetamide
ethyl 4-[9-hydroxy-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidine-1-carboxylate
N-[1-(1-cyclohexanecarbonylpiperidin-4-yl)-2-(3-methoxyphenyl)ethyl]-N,1-dimethyl-1H-pyrazole-3-carboxamide
2-{[4-(3-chlorophenyl)-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-methyl-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-(pyrimidin-4-ylmethyl)acetamide
4-oxo-4-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]butane-1-sulfonamide
N5-cyclooctyl-N3,N3-diethyl-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-{2-[1-(furan-2-ylmethyl)piperidin-3-yl]ethyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-(ethylamino)-N-[1-(4-fluorophenyl)-2-methylpropan-2-yl]pyrimidine-5-carboxamide
(3S,9aR)-3-(cyclohexylmethyl)-8-(2,5-dimethylbenzenesulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
[(3R,4R)-1-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
(2S,4S)-4-amino-1-(6-methylpyridine-2-carbonyl)pyrrolidine-2-carboxylic acid
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-2-{4-[(6-methylpyridin-2-yl)methyl]morpholin-3-yl}acetamide
5-(cyclooctylamino)-1-ethyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-4-sulfamoylbenzamide
(2S,4S)-4-amino-1-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylacetamide
6-{8-[2-(dimethylamino)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecane-2-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(3-methylpyridin-2-yl)-4-{[1-(propan-2-yl)-1H-pyrrol-3-yl]methyl}piperazine
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-[(3R,4S)-1-(oxan-4-yl)-4-propylpyrrolidin-3-yl]propanamide
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(thiophene-3-carbonyl)pyrrolidin-3-amine
3-bromo-5-(cyclopentylsulfamoyl)benzoic acid
4-cyclopentyl-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(5-ethylpyridin-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-cyclopropyl-1-[1-(1H-indole-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
methyl (2S)-1-{1-[4-(3-phenylpropanamido)phenyl]piperidin-4-yl}pyrrolidine-2-carboxylate
N-[(3S,5S)-1-[(3-ethenylphenyl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
5-{3-[3-(2-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl}-5-(thiophen-2-ylmethyl)pyrrolidin-2-one
N-cyclopentyl-3-{5-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-[5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
(3R,4S)-1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-cyclopropylpyrrolidin-3-amine
2-amino-N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-ethylpiperazine
[(3R,4S)-4-(morpholin-4-ylmethyl)-1-{[2-(trifluoromethoxy)phenyl]methyl}pyrrolidin-3-yl]methanol
2-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]pyrrolidin-2-yl}-1,3-benzothiazole
N-[(3R,4S)-1-(carbamoylmethyl)-4-cyclopropylpyrrolidin-3-yl]-3-(3-chloro-1H-1,2,4-triazol-5-yl)propanamide
5,7-dimethyl-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
4-ethoxy-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]pyrimidin-2-amine
N-(1-{[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)carbamoyl]methyl}-1H-pyrazol-4-yl)furan-2-carboxamide
4-{1-methyl-4-[3-(propoxymethyl)pyrrolidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
3-(5-chloro-1-methyl-4-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-ylmethyl}-1H-pyrazol-3-yl)-5-methyl-1,2-oxazole
N-methyl-N-[(3-methyloxetan-3-yl)methyl]-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-[(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)methyl]benzoic acid
2-methyl-3-{3-[2-methyl-6-(trifluoromethyl)pyridin-3-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyrazine
2-(2-hydroxyethyl)-8-[5-(trifluoromethyl)pyridin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
2-({cyclopropyl[(2-ethoxyphenyl)methyl]amino}methyl)-6-methoxyphenol