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7-(3,6-dimethylpyrazin-2-yl)-4-(2-methyloxolane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
9-[2-(4-fluorophenyl)acetyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(2,6-difluoro-3-methylphenyl)methyl]-1-[2-(dimethylamino)ethyl]-6-oxopiperidine-3-carboxamide
1-[2-ethoxy-5-(trifluoromethyl)phenyl]-3-methyl-3-(1,2-oxazol-3-ylmethyl)urea
1-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
3-{[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})amino}-2,2-dimethylpropan-1-ol
2-[methyl(pyridin-4-ylmethyl)amino]-1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}ethan-1-one
N-[1-(morpholin-4-ylmethyl)cyclopentyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
N-[1-(4-chlorophenyl)ethyl]-3-[(4-fluorophenyl)methyl]-1,2-oxazole-5-carboxamide
1-(1-benzylpiperidin-4-yl)-3-(1-propyl-1H-1,2,4-triazol-3-yl)urea
N-{2-[5-(3-fluoro-4-methylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}acetamide
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-methyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
(1S,4S)-5-(3-hydroxypropyl)-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
3-[(3S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-[(4-methoxyphenyl)methyl]propanamide
3-cyclopropyl-N-(1,3-dihydro-2-benzofuran-5-yl)-1H-pyrazole-5-carboxamide
N-(1-hydroxybutan-2-yl)-4-methyl-N-(thiophen-2-ylmethyl)pyridine-3-carboxamide
2-[3-benzyl-1-(3-methylphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-cyclopropylacetamide
(4S)-1-[1-(4-chlorophenyl)piperidin-4-yl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
1-[(4-fluorophenyl)methyl]-4-(2-methoxypyridine-3-carbonyl)-2-(propan-2-yl)-1,4-diazepane
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(pent-4-enoyl)pyrrolidin-3-yl]-1-methyl-1H-imidazole-5-carboxamide
methyl 1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine-4-carboxylate
N-(1-hydroxybutan-2-yl)-2-methyl-N-(thiophen-3-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
9-methoxy-7-(4-methylphenyl)-4-(1H-pyrrol-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[3-(1H-imidazol-1-yl)propyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
1-butyl-3-cyclopropyl-5-(2,4-dimethoxyphenyl)-1H-1,2,4-triazole
7-methyl-3-[3-(5-methylfuran-2-yl)butyl]-3,7,11-triazaspiro[5.6]dodecan-12-one
1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-ol
4-phenyl-2-{4-[(2R)-pyrrolidine-2-carbonyl]piperazin-1-yl}pyrimidine
1-(4-methylphenyl)-4-(3,4,7-trimethyl-1H-indole-2-carbonyl)piperazin-2-one
3-(2-chlorophenyl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}propanamide
4-[(1E)-3-[7-(1-hydroxy-2-phenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]prop-1-en-1-yl]-2-methoxyphenol
3-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}-1H-pyrazole
2-ethyl-9-(1H-imidazol-2-ylmethyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
1-(2,3-dihydro-1H-inden-2-yl)-2-(2,2-dimethyloxan-4-yl)-1H-imidazole
N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2,7,8-trimethylquinoline-4-carboxamide
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
3-(4-chlorobenzoyl)-1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidine
(3S,5S)-1-methyl-5-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]pyrrolidin-3-amine
2-[2-(4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperazin-1-yl)ethoxy]ethan-1-ol
2-[(2-methylphenyl)sulfanyl]-N-[1-(pyrimidin-4-yl)ethyl]acetamide
1-[(3-fluorophenyl)methyl]-N-[(5-methylthiophen-2-yl)methyl]-6-oxopiperidine-3-carboxamide
2-phenyl-1-[1-(3-phenyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]ethan-1-one
methyl 3-(furan-3-amido)-5-({[4-(morpholin-4-yl)phenyl]formamido}methyl)benzoate
4-{3-[2-(1-phenylethyl)-1H-imidazol-1-yl]propyl}morpholine
N3-cycloheptyl-1-cyclopropyl-N5-[(1R)-1-(4-methoxyphenyl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2,6-dimethyl-4-{[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl}phenyl acetate
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
(3R,4S)-4-(4-methoxyphenyl)-1-[2-(pyrrolidin-1-yl)benzoyl]pyrrolidin-3-amine
2-(2H-1,2,3-benzotriazol-2-yl)-N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)acetamide
1-methyl-N-{[8-(3-methylbut-2-en-1-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-6-oxo-1,6-dihydropyridazine-3-carboxamide