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N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-3-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-(2-methoxyethoxy)ethan-1-one
2-(2-ethoxyphenyl)-2-{methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}acetic acid
4-{[2-(3-chloro-5-fluoro-4-methoxyphenyl)-1H-imidazol-1-yl]methyl}pyridine
N-cyclopropyl-4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]sulfamoyl}benzamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]quinoxalin-2-amine
5-(3-methylbutyl)-5-{1-[(2-methylphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
3-(4-fluorophenyl)-4-[3-(4-hydroxyphenyl)-1H-pyrazole-5-carbonyl]piperazin-2-one
N-(2-hydroxypropyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(3-methylphenoxy)piperidine
[3-(3-methylbut-2-en-1-yl)-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]piperidin-3-yl]methanol
2-({2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}amino)propan-1-ol
1-{1-[(3-fluorophenyl)methyl]piperidin-3-yl}-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
4-methoxy-2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
1-[(2,4-dimethoxyphenyl)methyl]-5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazole
6-({[4-(dimethylamino)-1-methylpiperidin-4-yl]methyl}amino)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}azetidin-3-amine
1-(4-cyclopentyl-1,4-diazepan-1-yl)-2-hydroxy-2-(4-methoxyphenyl)ethan-1-one
2-[4-(2,4-dimethoxyphenyl)-6-methylpyrimidin-2-yl]phenol
5-chloro-3-fluoro-2-(2-{[(3S)-3-fluoropyrrolidin-1-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)pyridine
2-{4-[(dimethylamino)methyl]phenyl}-N-ethylpyrimidin-4-amine
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
N-{2-[4-(dimethylamino)phenyl]ethyl}-2,6-dimethylpyridine-4-carboxamide
2-[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-indazol-3-yl)acetamide
4-(2-methoxyethoxy)-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidine
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
2-(1-ethylpiperidin-4-yl)-1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]ethan-1-one
8-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aR,5S,6S,7aS)-2-[(1-methyl-1H-indol-2-yl)methyl]-octahydro-1H-isoindole-5,6-diol
1-[(2,6-dimethoxyphenyl)methyl]-3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
methyl 1-(2-methoxyethoxy)-2-oxo-8-[2-(4-phenylphenyl)acetyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
(3S,4S)-4-cyclopropyl-1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}pyrrolidine-3-carboxylic acid
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(morpholin-4-yl)acetamide
2-chloro-3-(1H-imidazol-2-yl)-9-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
2-[methyl(oxan-4-ylmethyl)amino]-2-(4-methylphenyl)acetic acid
4-methoxy-2-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]phenol
2-(1-ethyl-1H-pyrazole-4-carbonyl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
1-({4-methyl-5-[1-(1,3-thiazol-4-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
N-[2-(2-methyl-1H-indol-3-yl)ethyl]-3-(morpholin-4-yl)benzamide
3-{2-[methyl(2-phenylethyl)amino]ethyl}-8-(1-methylcyclopropanecarbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(3S,4R)-1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
2-methyl-6-(5-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}-3-(3-methylbutyl)-1H-1,2,4-triazol-1-yl)pyridine
3-(3-hydroxy-3-methylbutyl)-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]benzamide
3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-1-(5-oxo-1-propylpyrrolidin-3-yl)urea
2-(1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
2-(cyclohex-1-en-1-yl)-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]acetamide
4-methoxy-N-({1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
2-[({[1-(piperidin-1-yl)cyclohexyl]methyl}amino)methyl]-4-(pyridin-2-yl)phenol