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2-(dimethylamino)-4-methyl-N-[2-(4-phenylpyrimidin-2-yl)ethyl]pyrimidine-5-carboxamide
3-{2-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-4-yl]-2-oxoethyl}-5,5-dimethylimidazolidine-2,4-dione
1-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazole
2-[3-fluoro-5-(trifluoromethyl)phenyl]-2-[methyl(1,2-oxazol-3-ylmethyl)amino]acetic acid
3-(5-amino-1H-1,2,4-triazol-3-yl)-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]propanamide
(4aS,8aR)-6-[(8-chloroquinolin-2-yl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2,1-benzoxazole-3-carboxamide
1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-4-(pyridin-4-yl)piperazine
4-[butyl({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl})amino]butan-1-ol
6-[2-(1H-pyrazol-1-yl)ethyl]-2-[4-(thiomorpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
1-ethyl-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
(2S,4S)-N-ethyl-4-[(5-methyl-1,3,4-thiadiazol-2-yl)amino]-1-[(5-methylfuran-2-yl)methyl]pyrrolidine-2-carboxamide
N-benzyl-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(1-methylpiperidin-4-yl)-2-(morpholin-2-yl)-N-(pyridin-4-ylmethyl)acetamide
1-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-4-(1H-pyrazol-1-ylmethyl)piperidine
methyl 2-(4-acetamidophenyl)-5-methoxybenzoate
N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
N-[4-(1H-pyrazol-1-yl)phenyl]-1-[2-(pyrrolidin-1-yl)acetyl]piperidine-2-carboxamide
3-ethyl-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
1-{6-hydroxy-4-[(2-methylnaphthalen-1-yl)methyl]-1,4-diazepan-1-yl}ethan-1-one
1-(2-methoxybenzoyl)-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperazine
(2S,4S)-1-[(3-chlorophenyl)methyl]-N,N-diethyl-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
2-{5-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-pyrazol-3-yl}phenol
N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
1-butyl-4-(1H-pyrazole-4-carbonyl)piperazin-2-one
[(3R,4S)-1-{[2-(difluoromethoxy)phenyl]methyl}-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-(naphthalen-1-ylmethyl)benzamide
1-(1-cycloheptylpiperidin-4-yl)-N-(2-hydroxyethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
5-(2-methoxyphenoxymethyl)-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-1H-pyrazole-3-carboxamide
methyl 4-(4-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)benzoate
4-{4-[(3-methylthiophen-2-yl)methyl]piperazin-1-yl}-2-{[4-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
2-(ethylamino)-N,4-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-thiazole-5-carboxamide
methyl 3-[(3S,4R)-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-1-[(2-hydroxynaphthalen-1-yl)methyl]piperidin-3-yl]propanoate
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
9-(2-ethoxypropanoyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(1-methoxypropan-2-yl)-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidine
5-methoxy-1-methyl-2-{3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl}-1H-indole
6-methyl-3-[3-(pyrimidin-4-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-{[1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl]oxy}pyrimidine
2-[(2S,4R)-4-amino-2-(diethylcarbamoyl)pyrrolidin-1-yl]-N-methylpyridine-3-carboxamide
3-[(3R,4S)-1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
2-(1-{4-[(diethylamino)methyl]-5-ethylfuran-2-amido}cyclohexyl)acetic acid
4-methyl-6-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-1,4-oxazepane
{[2,4-bis(prop-2-en-1-yloxy)phenyl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
8-(3-ethyl-1H-indole-2-carbonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}(methyl)[1-(3-methylpyridin-2-yl)propan-2-yl]amine
2-methyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-[1-(4-acetylbenzoyl)piperidin-4-yl]-5-[(2-chlorophenyl)methyl]imidazolidine-2,4-dione