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1-benzoyl-4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-[2-(1H-indol-1-yl)ethyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
(1S,5R)-6-[(3,5-dichloropyridin-4-yl)methyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-chloro-4-{[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]oxy}-N-[2-(dimethylamino)ethyl]benzamide
3-cyclopropanecarbonyl-9-{[3-(propan-2-yloxy)phenyl]methyl}-3,9-diazaspiro[5.5]undecane
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(oxan-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[4-(4-{[(1-benzyl-1H-pyrazol-4-yl)methyl]amino}piperidin-1-yl)phenyl]-2-(3-fluorophenyl)acetamide
1-methyl-N-({5-methyl-2-[2-(oxolane-2-amido)phenyl]-1,3-oxazol-4-yl}methyl)-3-propyl-1H-pyrazole-5-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]propan-1-one
8-(ethanesulfonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(pyrazine-2-carbonyl)piperidin-4-yl]propanamide
N-({8-[(2-methoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1-methyl-1H-pyrazole-3-carboxamide
6,7-dimethoxy-2-(1H-1,2,3-triazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline
(2E)-1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-3-(furan-2-yl)prop-2-en-1-one
N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
1-[3-(cyclooctylcarbamoyl)propanoyl]piperidine-4-carboxylic acid
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-4-methoxypyrimidin-2-amine
1-[2-(pyrrolidin-1-yl)benzoyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-[2-(4-fluorophenyl)ethyl]-N-({2-[3-(hydroxymethyl)piperidin-1-yl]-7-methoxyquinolin-3-yl}methyl)thiophene-2-carboxamide
5-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-3-[(4-fluorophenyl)methyl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
2-(1H-1,3-benzodiazol-1-yl)-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]propanamide
(2R,3S,6R)-5-(1H-1,2,3-benzotriazole-5-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-ethoxy-5-[2-(3-fluorophenoxymethyl)pyrimidin-4-yl]benzoic acid
3-[2-(dimethylamino)ethyl]-1-ethyl-8-[(9-ethyl-9H-carbazol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[2-(1H-imidazol-4-yl)ethyl]-8-[(6-methylpyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(dimethylamino)-2-(3-fluorophenyl)-N-(2-methoxyethyl)-N-(1-methylpiperidin-4-yl)acetamide
2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(4-methylpentanoyl)-2,7-diazaspiro[4.5]decan-6-one
3-{5-[(2r,4r)-6,8-dioxo-5,7-diazaspiro[3.4]octane-2-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
2-ethyl-N,4-dimethyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1,3-thiazole-5-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,1-dimethyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
2-(2-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}ethyl)-1H-1,3-benzodiazole
N-[2-(dimethylamino)ethyl]-N-(oxolan-2-ylmethyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
3-(3-hydroxy-3-methylbutyl)-N-{1-oxaspiro[4.5]decan-3-yl}benzamide
N-[2-(5-methylfuran-2-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2,2-dimethylpropan-1-one
4-[4-(dimethyl-1,2-oxazole-4-carbonyl)piperazin-1-yl]quinazoline
2-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-methyl-N-(quinolin-2-ylmethyl)acetamide
2-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}quinoline
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2,2,3-trimethylbut-3-en-1-one
{1-[1-(2,3-dihydro-1H-inden-4-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]cyclopropyl}methanol
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(4-propanoylphenoxy)acetamide
N-(2-{[2-(2-aminoethyl)quinazolin-4-yl]amino}ethyl)-4-fluorobenzamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-2-phenylpyrimidine-5-carboxamide
(4aR,8aS)-6-[(2,4-dimethoxy-3-methylphenyl)methyl]-1-[2-(2-fluorophenyl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-(2,3-dihydro-1H-inden-2-yl)-3-(2-hydroxyphenyl)-3-(3-hydroxyphenyl)propanamide
(3S,4R)-1-(2,1,3-benzothiadiazol-4-ylmethyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
methyl 1-ethoxy-8-[(2-ethoxyphenyl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
(2S)-2-hydroxy-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-3-phenylpropanamide