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2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[2-(1,3-thiazol-4-yl)ethyl]acetamide
5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-4-methylpyrimidin-2-amine
5-[(4-fluorophenyl)methyl]-5-(piperidin-4-yl)-3-(1,3-thiazol-5-ylmethyl)imidazolidine-2,4-dione
5-fluoro-2-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
2-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-5-methylpyrazine
1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(thiophene-2-carbonyl)piperidine
N-[(2R,3R)-1'-[2-(cyclohex-1-en-1-yl)acetyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
N-ethyl-N-[2-(pyrrolidin-1-yl)ethyl]piperidin-4-amine
N5-cycloheptyl-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
5-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)pyrrolidin-2-yl]-N-(pyridin-3-yl)thiophene-2-carboxamide
4-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}-7-hydroxy-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
1-(4-ethylpiperazin-1-yl)-3-[2-methoxy-4-({methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
(2S,4S)-N-ethyl-1-(furan-2-ylmethyl)-4-[(2E)-3-phenylprop-2-enamido]pyrrolidine-2-carboxamide
1-(3-phenylpropyl)-5-(pyridine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
5-cyclobutanecarbonyl-1'-[(5-methylthiophen-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)pyridine-3-carboxamide
(2R,4S)-4-hydroxy-1-[4-(1H-indol-3-yl)butanoyl]piperidine-2-carboxylic acid
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-{3-[(4-fluorophenyl)formamido]propanamido}acetic acid
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)acetamide
[(1-cyclopentylpiperidin-4-yl)methyl][(1-methyl-1H-pyrazol-4-yl)methyl](pyridin-3-ylmethyl)amine
2-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1-methyl-5-phenyl-1H-pyrrole
1-[3-(1,4-diazepane-1-carbonyl)benzenesulfonyl]piperidin-3-ol
(3aS,7aR)-5-methyl-2-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
3-[2-(4-fluorophenyl)piperidine-1-carbonyl]-1-methyl-1,4-dihydroquinolin-4-one
N-[1-(pyrazin-2-yl)propan-2-yl]-4-(1H-pyrazol-3-yl)benzamide
6-{2-oxa-7-azaspiro[4.5]decan-7-ylmethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)benzoic acid
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
3-{2-[3-oxo-3-(pyrrolidin-1-yl)propyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}propanamide
2-{2-oxo-8-[(3R)-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetic acid
1-(azocan-1-yl)-3-[2-methoxy-4-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
4-hydroxy-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-2-phenylpyrimidine-5-carboxamide
1-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
1-(pyridin-3-ylmethyl)-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-1,4-diazepane
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-ethoxyacetamide
2-methyl-5-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]-1,3-benzothiazole
(2S,4S)-N-ethyl-1-(oxan-4-yl)-4-[3-(pyridin-3-yl)propanamido]pyrrolidine-2-carboxamide
6-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methyl-1,3-thiazole-5-carboxamide
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1,1-dioxo-1λ6-thiolane-3-carboxamide
5-(2-fluorophenoxymethyl)-N-methyl-N-[(1-methylpiperidin-4-yl)methyl]-1H-pyrazole-3-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
(2E)-N-cyclopropyl-3-(3-fluorophenyl)-N-({4-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)prop-2-enamide
N-[(1-{2-[(1R,4S)-2-azabicyclo[2.2.1]heptan-2-yl]ethyl}-1,2,5,6-tetrahydropyridin-3-yl)methyl]acetamide
3-[({1-[(3-fluoro-2,4-dimethylphenyl)methyl]piperidin-4-yl}oxy)methyl]pyridine
5-{1-[4-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}-3-(propan-2-yl)-1,2,4-oxadiazole
2-(methylsulfanyl)-4-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidine
(1-{[methyl({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})amino]methyl}cyclopropyl)methanol
5,7-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-N-(2-methylpropyl)-2-oxoacetamide