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2-(adamantan-1-yl)-4-hydroxy-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]pyrimidine-5-carboxamide
2-{[4-(2-fluorophenyl)-5-[(propan-2-yloxy)methyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamide
2-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-6-(trifluoromethyl)pyridine-3-carboxamide
3,5-dimethyl-1-[1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidin-3-yl]-1H-pyrazole
N-[(4-methylphenyl)methyl]-5-(2-methylpiperidine-1-carbonyl)-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-(2-propoxyacetyl)piperazin-2-one
3-methyl-3-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1-[4-(propylsulfamoyl)phenyl]urea
1-(3-methoxyphenyl)-6-methyl-4-[2-(trifluoromethyl)benzoyl]piperazin-2-one
5-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]-2,1,3-benzoxadiazol-1-ium-1-olate
(8R,9aS)-8-hydroxy-2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
N'-(3,5-dimethylphenyl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]propanediamide
(1R,5R)-6-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-{1-[(2-fluorophenyl)methyl]-4-(1H-indol-2-ylmethyl)piperazin-2-yl}ethan-1-ol
5-{[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
N-cyclopropyl-1-{1-[6-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}piperidine-3-carboxamide
3-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-4-yl)-N-(pyridin-3-ylmethyl)propanamide
1-methanesulfonyl-4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazine
2-[3,5-dimethyl-4-(2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamido)-1H-pyrazol-1-yl]acetic acid
({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
(adamantan-1-ylmethyl)({[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
N-[2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]pyridine-4-carboxamide
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-(2-methoxyethoxy)ethan-1-one
6-[(diethylamino)methyl]-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[(2R)-pyrrolidin-2-ylmethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
4-(4-methoxybutyl)-N-(3-methylphenyl)piperazine-1-carboxamide
7-(1,3-benzothiazol-2-yl)-9-(oxolan-3-yloxy)-4-[4-(trifluoromethyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-(3-chlorophenyl)-4-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}amine
2-{5-[(1-methyl-1H-imidazol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-propyl-1H-imidazole
1,3-dimethyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-(2-amino-1,3-benzothiazole-5-carbonyl)-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
2-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)-1-(prop-2-en-1-yl)-1H-1,3-benzodiazole
N-({1-[(2,6-dimethoxyphenyl)methyl]piperidin-3-yl}methyl)methanesulfonamide
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-2-ethylpyrimidine-5-carboxamide
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(naphthalene-1-carbonyl)piperidine
(2S,4R)-N-[(2-chlorophenyl)methyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
2-(1,3-benzoxazol-2-yl)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]acetamide
2-(4-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)pyrazine
N-[1-(4-methyl-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]-2-(pyridin-2-ylsulfanyl)acetamide
(3aS,6aR)-3-[2-(pyridin-2-yl)ethyl]-5-(quinolin-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[2-oxo-2-(4-phenylpiperidin-1-yl)ethyl]-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidine-2,5-dione
1-(2-methoxy-4-{[methyl(2-phenoxyethyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
N-(7-{6-azabicyclo[3.2.1]octane-6-carbonyl}-2-ethyl-1-(pyridin-3-ylmethyl)-1H-1,3-benzodiazol-5-yl)acetamide
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-(cyclopropylmethyl)-5-[2-(methylamino)-1,3-thiazole-4-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carbonitrile
6-cyclopentyl-2-methoxy-3-{[(propan-2-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
5-{1-[(2,5-dimethoxyphenyl)methyl]piperidin-4-yl}-5-(3-phenylpropyl)imidazolidine-2,4-dione
ethyl(2-{4-[3-(1H-pyrazol-3-yl)phenyl]phenoxy}ethyl)amine