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1-(2-{[cyclohexyl(methyl)amino]methyl}phenyl)-3-ethyl-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]urea
[(4-fluoro-2-methoxyphenyl)methyl](methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
2-[4-(3,4-dimethoxybenzenesulfonyl)morpholin-3-yl]acetic acid
N-methyl-N-[(1R)-1-(naphthalen-1-yl)ethyl]-6-(piperidin-4-yl)pyrimidin-4-amine
2-[(4-chlorophenyl)methyl]-N-[2-(propan-2-yloxy)ethyl]-1,3-benzoxazole-5-carboxamide
5-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-pyrazol-1-yl)propan-1-one
6-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-5,6-dihydro-1,6-naphthyridin-5-one
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
[9-(pyridin-3-ylmethyl)-3-(pyridine-4-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-(5-ethylthiophene-3-carbonyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
3-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chloro-2-methylphenyl)urea
3-amino-2-methyl-1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
N-cyclohexyl-3-{[5-(methoxymethyl)thiophen-2-yl]formamido}propanamide
(2S,4R)-4-[(2,3-dihydro-1H-inden-2-yl)amino]-N-ethyl-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide
N-methyl-2-phenyl-N-(quinolin-4-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
N-(1H-imidazol-2-ylmethyl)-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide
1-[3-({[2-(cyclohex-1-en-1-yl)ethyl]amino}methyl)phenoxy]-3-(4-ethylpiperazin-1-yl)propan-2-ol
N-[(2R,3R)-1'-(3-methylbenzoyl)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-(4-{[1-(2,5-difluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenyl)acetamide
5-ethyl-5-[3-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-3-oxopropyl]pyrrolidin-2-one
2,5-dioxo-6-[2-(4,5,6,7-tetrahydro-1H-indazol-3-yl)ethyl]-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-amino-6-(4-hydroxyphenyl)-4-[1-(pyridin-3-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
N-[2-(4-chlorophenyl)ethyl]-2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
benzyl(butyl){[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
(2R,6S)-4-{2-[(4-benzylpiperazin-1-yl)methyl]-1,3-oxazole-4-carbonyl}-2,6-dimethylmorpholine
4-(2,3-dihydro-1-benzofuran-7-yl)-6-(propan-2-yloxy)pyrimidin-2-amine
1-(1,3-benzothiazole-6-carbonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-(2-ethoxyethyl)-5-methylpiperidin-2-one
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-[3-(pyridin-2-yl)azetidin-1-yl]butan-1-one
(5S,9aS,9bS)-5-(1-ethyl-5-methyl-1H-pyrazol-4-yl)-2-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-3-(1,2-oxazinan-2-yl)propanamide
1-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
7-[4-(diethylamino)benzoyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-6-methyl-1-(propan-2-yl)-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
3,6-dimethyl-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
7-(cyclohexylmethyl)-2-(1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-(cyclohex-1-en-1-ylmethyl)-3-(2,5-dioxoimidazolidin-4-yl)propanamide
{[4-({1-[5-(4-methoxyphenyl)furan-2-carbonyl]piperidin-4-yl}oxy)phenyl]methyl}(methyl)(quinolin-6-ylmethyl)amine
N-[1-(2-phenylethyl)piperidin-3-yl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
(2E)-3-(2-chlorophenyl)-1-{4-[4-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]piperidin-1-yl}prop-2-en-1-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-1,3-oxazole-4-carboxamide
dimethyl({[(1R,5S,6S)-3-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
5-[(2-fluorophenyl)methyl]-5-[1-(3-phenylpropyl)piperidin-4-yl]imidazolidine-2,4-dione
N-{[5-(3-chlorophenyl)furan-2-yl]methyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]piperidin-4-amine
2-methyl-3-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)phenol
1-{2-[2-(pyridin-2-yl)ethoxy]phenyl}-3-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}urea