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2-acetyl-8-(3-hydroxy-2-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(3-acetyl-1H-indol-1-yl)-1-(1,2,3,6-tetrahydropyridin-1-yl)butan-1-one
4-(4-chlorophenyl)-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]butanamide
N-[(3-methoxyphenyl)methyl]-3-[1-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)piperidin-3-yl]propanamide
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}morpholine-2-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(2-methyl-1,3-oxazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(1-ethyl-1H-indazol-3-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
4-[1-(1-methoxybutan-2-yl)-4-phenyl-1H-imidazol-5-yl]-2,1,3-benzoxadiazole
4-methyl-1-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pentane-1,2-dione
6-(cyclohexylamino)-2-methylheptan-2-ol
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}pyrimidin-4-amine
N-[3-(furan-2-yl)phenyl]-1-(pyridin-3-ylmethyl)piperidine-4-carboxamide
(3S,4S)-1-(6-chloropyridazin-3-yl)-4-(naphthalen-2-yl)piperidin-3-ol
1,2-dimethyl-N-(5-oxo-1-phenylpyrrolidin-3-yl)-1H-imidazole-4-sulfonamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-5-methylhexanamide
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]acetamide
N-(3-hydroxypropyl)-1-methyl-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrrole-2-carboxamide
1-[2-(dimethylamino)ethyl]-4-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}pyrrolidin-2-one
3-(4-methoxyphenyl)-1-(4-methylpiperazin-1-yl)-3-phenylpropan-1-one
2-[4-(azocan-1-yl)-5-methylthieno[2,3-d]pyrimidine-6-carbonyl]-2-azabicyclo[2.2.1]heptane
3-{[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-5-(2-methylpropyl)-1,2,4-oxadiazole
8-(4-aminopyridine-2-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(2,3-dihydro-1H-inden-1-yl)-1-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
(3S,4S)-4-cyclopropyl-1-(2,3-dihydro-1H-indene-5-carbonyl)pyrrolidine-3-carboxylic acid
N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
{4-[(5-{[6-(dimethylamino)pyridin-3-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]-1-methylpiperazin-2-yl}methanol
3-[(2R,3R,6R)-5-(3-fluoro-4-methoxybenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
5-methyl-N-[3-(methylsulfanyl)propyl]-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2-[(4-fluorophenyl)methyl]-4-(3-methylfuran-2-carbonyl)morpholine
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-(3-methylbenzoyl)piperidine
4-(2-methoxyphenyl)-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]benzamide
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2,3-dihydro-1-benzofuran-2-carboxamide
N-[2-(4-phenylpiperidin-1-yl)ethyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
1-(2-hydroxyethyl)-N-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carboxamide
3-methyl-6-{2-[(4-methylpiperazin-1-yl)methyl]phenoxy}pyridazine
ethyl 2-[N-methyl-1-(3-methyl-5-propyl-1-benzofuran-2-yl)formamido]acetate
[(1,5-dimethyl-1H-indazol-3-yl)methyl][4-(1H-pyrazol-1-yl)butan-2-yl]amine
N-(1-{7-[(4-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
5-methyl-N-(1,2-oxazol-3-ylmethyl)-4-{[(4-phenyloxan-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
4,7,8-trimethyl-2-(pyrimidin-5-yl)quinoline
1-methyl-N-{[8-(thiophen-3-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1H-pyrazole-5-carboxamide
4-[(2,4-dimethylphenyl)methyl]-9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-yl]ethan-1-one
9-(5-hydroxypyrazine-2-carbonyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-4-[(2-methyl-1H-imidazol-4-yl)methyl]-1,4-diazepan-6-ol
1-[(2,3-difluorophenyl)methyl]-4-[1-(1,2,3-thiadiazole-4-carbonyl)pyrrolidin-3-yl]piperidine
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-4-(piperidin-3-yl)benzamide