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2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-fluorophenyl)methyl]-N-methylacetamide
[(2S,4R,5R)-5-(4-chlorophenyl)-1-ethyl-4-({[(4-methoxyphenyl)methyl]amino}methyl)-2-methylpyrrolidin-2-yl]methanol
N-[(5-methylthiophen-2-yl)methyl]-3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-(prop-2-en-1-yl)propanamide
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidine
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-4-(piperidin-3-yl)benzamide
1-methyl-3-(2-methyl-1,3-benzothiazol-5-yl)-1-[1-(4-methylpyridin-2-yl)propan-2-yl]urea
3-benzyl-1-(3-methoxypropyl)-8-[3-(5-methylfuran-2-yl)butyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-phenoxy-N-{1-[1-(pyridine-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
1-(3-{[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-oxopiperidin-1-yl)acetamide
N-(1-{1-[2-(4-methoxyphenoxy)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
N'-(3-chloro-4-fluorophenyl)-N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]butanediamide
2-ethyl-8-[2-(pyridin-2-yl)pyrimidine-5-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
2-butoxy-1-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one
N-{3H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(3-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
4-[2-(2-phenylethyl)-3H-imidazo[4,5-b]pyridin-3-yl]-1-(thiophen-3-ylmethyl)piperidine
3-{ethyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}-1λ6-thiolane-1,1-dione
2-(2-chloro-4-{[2-(1,3-thiazol-2-yl)piperidin-1-yl]methyl}phenoxy)acetamide
N-(4-methyl-1-propyl-1H-pyrazol-5-yl)-2-[4-(3-methylpyrazin-2-yl)-1H-pyrazol-1-yl]acetamide
1-cyclohexyl-N-[2-(3-fluorophenyl)-2-hydroxyethyl]piperidine-4-carboxamide
1-[(4-fluorophenyl)methyl]-4-({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amino)pyrrolidin-2-one
2-[3-(2,5-dimethylfuran-3-yl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
(2R,6S)-2,6-dimethyl-4-[5-(piperidin-1-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carbonyl]morpholine
3-ethyl-4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperazin-2-one
5,7-dimethyl-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]pyrido[2,3-d]pyrimidin-4-amine
4-(hydroxymethyl)-5-methyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
(5S,9aS,9bS)-5-(5-chloro-2,3-dimethoxyphenyl)-2-cyclopentyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
methyl (2S,4R)-4-(5-chloro-3-methyl-1H-indole-2-amido)-1-[(3-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
1-(1H-1,3-benzodiazol-2-ylmethyl)-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
2-benzyl-5-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,3-benzoxazole
3-(pyrrolidin-1-yl)-6-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyridazine
N-[(2-chloro-6-fluorophenyl)methyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
(2S,5R)-1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,5-dimethylpiperazine
1-(cyclohexylmethyl)-N,N-dimethyl-5-[(1,2-oxazol-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
5-[3-chloro-5-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxymethyl]-3-cyclopropyl-1,2,4-oxadiazole
1-(1'-{[2-(ethylamino)pyrimidin-5-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)propan-1-one
ethyl 4-(5-ethyl-2-methylpyrimidin-4-yl)piperazine-1-carboxylate
N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}imidazo[1,2-a]pyridine-6-carboxamide
2-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
7-(5-chloropyridin-2-yl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-N-(naphthalen-1-yl)piperidine-1-carboxamide
1-ethyl-5-(4-propylpyrimidine-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-(2-methoxyethyl)-3-(1,2,3-thiadiazol-5-yl)-1-(thiophen-2-ylmethyl)urea
{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[4-(trifluoromethyl)phenyl]methyl}amine
N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-(3-methylthiophene-2-carbonyl)piperidine
8-(furan-2-ylmethyl)-3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)pyridine
(3R,4R)-4-cyclobutyl-3-methyl-1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]piperidin-4-ol